Structure-Based Evolution of Subtype-Selective Neurotensin Receptor Ligands
Subtype-selective agonists of the neurotensin receptor NTS2 represent a promising option for the treatment of neuropathic pain, as NTS2 is involved in the mediation of μ-opioid-independent anti-nociceptive effects. Based on the crystal structure of the subtype NTS1 and previous structure–activity re...
Main Authors: | , , , , , , |
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Format: | Online |
Language: | English |
Published: |
Blackwell Publishing Ltd
2014
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Online Access: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4234217/ |