Structural Probing of Off-Target G Protein-Coupled Receptor Activities within a Series of Adenosine/Adenine Congeners

by Paoletta, Silvia, Tosh, Dilip K., Salvemini, Daniela, Jacobson, Kenneth A.
Published 2014

Polyamidoamine (PAMAM) dendrimer conjugate specifically activates the A3 adenosine receptor to improve post-ischemic/reperfusion function in isolated mouse hearts

by Wan, Tina C, Tosh, Dilip K, Du, Lili, Gizewski, Elizabeth T, Jacobson, Kenneth A, Auchampach, John A
Published 2011

John Daly Lecture: Structure-guided Drug Design for Adenosine and P2Y Receptors☆

by Jacobson, Kenneth A., Gao, Zhan-Guo, Paoletta, Silvia, Kiselev, Evgeny, Chakraborty, Saibal, Jayasekara, P. Suresh, Balasubramanian, Ramachandran, Tosh, Dilip K.
Published 2014

Purine (N)-Methanocarba Nucleoside Derivatives Lacking an Exocyclic Amine as Selective A3 Adenosine Receptor Agonists

by Tosh, Dilip K., Ciancetta, Antonella, Warnick, Eugene, O’Connor, Robert, Chen, Zhoumou, Gizewski, Elizabeth, Crane, Steven, Gao, Zhan-Guo, Auchampach, John A., Salvemini, Daniela, Jacobson, Kenneth A.
Published 2016

In Vivo Phenotypic Screening for Treating Chronic Neuropathic Pain: Modification of C2-Arylethynyl Group of Conformationally Constrained A3 Adenosine Receptor Agonists

by Tosh, Dilip K., Finley, Amanda, Paoletta, Silvia, Moss, Steven M., Gao, Zhan-Guo, Gizewski, Elizabeth T., Auchampach, John A., Salvemini, Daniela, Jacobson, Kenneth A.
Published 2014