A multicomponent reaction of 2-aminoimidazoles:
microwave-assisted synthesis of novel 5-aza-7-
deaza-adenines†‡

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A multicomponent reaction of 2-aminoimidazoles: microwave-assisted synthesis of novel 5-aza-7- deaza-adenines†‡

An efficient and highly selective multicomponent synthesis of 4-aminoimidazo[1,2-a][1,3,5]triazines, which are 5-aza-7-deaza-isosteres of adenine, was developed. The reaction of 2-aminoimidazoles, triethyl orthoformate and cyanamide under microwave irradiation proceeded regioselectively to provide...

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Bibliographic Details
Main Authors:	Lim, Felicia Phei Lin, Low, Szy Teng, Ho, Elvina Lee King, Halcovitch, Nathan R., Tiekink, Edward R. T. *, Dolzhenko, Anton V
Format:	Article
Language:	English
Published:	Royal Society of Chemistry 2017
Subjects:	QD Chemistry
Online Access:	http://eprints.sunway.edu.my/712/ http://eprints.sunway.edu.my/712/1/Tiekink%20A%20multicomponent%20RSC%20Adv%202017%20.pdf

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