Synthesis, in vitro evaluation, and radiolabeling of fluorinated puromycin analogues: potential candidates for PET imaging of protein synthesis

There is currently no ideal radiotracer for imaging protein synthesis rate (PSR) by positron emission tomography (PET). Existing fluorine-18 labelled amino acid-based radiotracers predominantly visualize amino acid transporter processes, and in many cases they are not incorporated into nascent prote...

Full description

Bibliographic Details
Main Authors: Betts, Helen M., Sephton, Selena Milicevic, Tong, Carmen, Awais, Ramla, Hill, Philip J., Perkins, A.C., Aigbirhio, Franklin I.
Format: Article
Published: American Chemical Society 2016
Subjects:
Online Access:https://eprints.nottingham.ac.uk/39443/