Structural elements of an NRPS cyclization domain and its intermodule docking domain

Epothilones are thiazole-containing natural products with anticancer activity that are biosynthesized by polyketide synthase (PKS)-nonribosomal peptide synthetase (NRPS) enzymes EpoA-F. A cyclization domain of EpoB (Cy) assembles the thiazole functionality from an acetyl group and l-cysteine via con...

Full description

Bibliographic Details
Main Authors: Dowling, Daniel P., Kung, Yan, Croft, Anna K., Taghizadeh, Koli, Kelly, Wendy L., Walsh, Christopher T., Drennan, Catherine L.
Format: Article
Published: National Academy of Sciences 2016
Subjects:
Online Access:https://eprints.nottingham.ac.uk/38671/