A practical drug discovery project at the undergraduate level

A practical drug discovery project at the undergraduate level

A practical drug discovery project for third-year undergraduates is described. No previous knowledge of medicinal chemistry is assumed. Initial lecture-workshops cover the basic principles; then students are asked to improve the profile of a weakly potent, poorly soluble PI3K inhibitor (1). Comp...

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Bibliographic Details
Main Authors: Fray, Michael J., Macdonald, Simon J.F., Baldwin, Ian R., Barton, Nick, Brown, Jack, Campbell, Ian B., Churcher, Ian, Coe, Diane M., Cooper, Anthony W.J., Craven, Andrew P., Fisher, Gail, Inglis, Graham G.A., Kelly, Henry A., Liddle, John, Maxwell, Aoife C., Patel, Vipulkumar K., Swanson, Stephen, Wellaway, Natalie
Format: Article
Published: Elsevier 2013
Subjects:
undergraduate research project
asthma
kinase
PI3K delta
thienopyrimidines
Online Access:https://eprints.nottingham.ac.uk/2292/

Internet

https://eprints.nottingham.ac.uk/2292/

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