Inhibition of OCTN2-mediated transport of carnitine by etoposide

OCTN2 is a bifunctional transporter that reabsorbs filtered carnitine in a sodium-dependent manner andsecretes organic cations into urine as a proton antiport mechanism. We hypothesized that inhibition of OCTN2 by anticancer drugs can influence carnitine resorption. OCTN2-mediated transport inhibiti...

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Bibliographic Details
Main Authors: Hu, C., Lancaster, C., Zuo, Zhili, Hu, S., Chen, Z., Rubnitz, J., Baker, S., Sparreboom, A.
Format: Journal Article
Published: American Association for Cancer Research 2013
Online Access:http://hdl.handle.net/20.500.11937/15970