Regio- and stereoselective synthesis of benzothiazolo-pyrimidinones via an NHC-catalyzed Mannich/lactamization domino reaction† †Electronic supplementary information (ESI) available. CCDC 1029497. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c4cc08594a

An NHC-catalyzed regio- and stereoselective Mannich/lactamization domino reaction of N-(benzothiazolyl)imines with α-chloroaldehydes has been developed.

Bibliographic Details
Main Authors: Ni, Qijian, Song, Xiaoxiao, Xiong, Jiawen, Raabe, Gerhard, Enders, Dieter
Format: Online
Language:English
Published: Royal Society of Chemistry 2015
Online Access:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4612130/