18F-FP-PEG2-β-Glu-RGD2: A Symmetric Integrin αvβ3-Targeting Radiotracer for Tumor PET Imaging

Radiolabeled cyclic arginine-glycine-aspartic (RGD) peptides can be used for noninvasive determination of integrin αvβ3 expression in tumors. In this study, we performed radiosynthesis and biological evaluation of a new 18F-labeled RGD homodimeric peptide with one 8-amino-3,6-dioxaoctanoic acid (PEG...

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Bibliographic Details
Main Authors: Hu, Kongzhen, Tang, Xiaolan, Tang, Ganghua, Yao, Shaobo, Yao, Baoguo, Wang, Hongliang, Nie, Dahong, Liang, Xiang, Tang, Caihua, He, Shanzhen
Format: Online
Language:English
Published: Public Library of Science 2015
Online Access:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4580323/