Ion channel drug discovery

Bibliographic Details
Main Authors: Cox, Brian (Author), Gosling, Martin (Author)
Format: Book
Language:English
Published: Cambridge : Royal Society of Chemistry , c2015
Series:RSC drug discovery series 39
Subjects:
Table of Contents:
  • 1. Ion channel drug discovery: a historical perspective
  • 2. High throughput screening
  • 3. Automated electrophysiology in ion channel drug discovery
  • 4. Structural understanding of ion channels in atomic detail
  • 5. Voltages-gated Sodium Channels: structure, function, and molecular pharmacology
  • 6. AMPA receptor positive allosteric modulators- a case history
  • 7. The discovery of novel inhaled ENaC blockers for the treatment of cystic fibrosis lung disease
  • 8. The therapeutic potential of small-molecule modulators of the cystic fibrosis transmembrane conductance regulator (CFTR) CI channel
  • 9. TRPV1 antagonism: from research to clinic
  • 10. Open access to the KCNQ channel: Retigabine and second generation M-current openers
  • 11. The therapeutic potential of hERG1 K channels for treating cancer and cardiac arrhythmias
  • 12. Does nature do Ion channel drug discovery better than us?
  • 13. Antibodies as Ion channel modulators
  • 14. Ion channel drug discovery: future perspectives