New horizons in predictive drug metabolism and pharmacokinetics

Bibliographic Details
Other Authors: Wilson, Alan G. E. , 1947- (Editor)
Format: Book
Language:English
Published: Cambridge : Royal Society of Chemistry c2016
Series:RSC drug discovery series no 49
Subjects:

MARC

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245 1 0 |a New horizons in predictive drug metabolism and pharmacokinetics   |c edited by Alan G. E. Wilson 
264 1 |a Cambridge :   |b Royal Society of Chemistry   |c c2016 
300 |a xxi, 422 pages :   |b illustration (some color) ;   |c 24 cm. 
336 |a text  |2 rdacontent 
337 |a unmediated  |2 rdamedia 
338 |a volume  |2 rdacarrier 
490 1 |a RSC drug discovery series   |v no 49 
504 |a Includes bibliographical references and index 
505 0 |a 1. How physicochemical properties of drugs affect their metabolism and clearance -- 2. Role of solubility, permeability and adsorption in drug discovery in development -- 3. Models for nonspecific binding and partitioning -- 4. Cytochrome P450 mediated drug metabolism -- 5. Non-cytochrome P450 enzymes and glucuronidation -- 6. Metabolite profiling -- 7. Application of humanised and other transgenic models to predict human responses to drugs -- 8. Stem cells and drug metabolism -- 9. Chemically reactive versus stable drug metabolites: Role in adverse drug reactions -- 10. Integrating metabolism and toxicity properties -- 11. Metabolomics-based approaches to determine drug metabolite profiles -- 12. Drug-drug ineteractions: regulatory and theoretical considerations, and an industrial perspective -- 13. Drug-drug interactions: Computational approaches -- 14. Induction of hepatic cytochrome P450 enzymes: Importance in drug development and toxicity -- 15. Current status and implications of transporters: QSAR analysis method to evaluate drug-drug interactions of human bile salt export pump (ABCB11/BSEP) and prediction of intrahepatic cholestasis risk -- 16. Formulation of optimizing bioavailability -- 17. Systems pharmacology modelling -- 18. Pharmacokinetic-pharmacodynamic modelling in drug development with special reference to oncology 
650 0 |a Drug development 
650 0 |a Drugs   |x Metabolism 
650 0 |a Pharmacokinetics 
650 2 |a Pharmaceutical Preparations   |x Metabolism 
650 2 2 |a Biopharmaceutics 
700 1 |a Wilson, Alan G. E. ,   |d 1947- ,   |e editor 
999 |a 1000169170   |b Book   |c OPEN SHELF (30 DAYS)   |e Tembila Campus