Pharmaceutical industry practices on genotoxic impurities

Bibliographic Details
Main Author: Lee, Heewon (Author)
Format: Book
Language:English
Published: Boca Raton, Florida : CRC Press c2015
Series:Chromatographic science series
Subjects:
Online Access:Cover image
Table of Contents:
  • 1. Overview of regulatory guidelines on impurities and genotoxic impurities
  • 2. Structural alerts for genotoxicity and carcinogenicity
  • 3. Acceptable exposure calculations for impurities and selected compounds from the carcinogenic potency database
  • 4. Genotoxic impurities from toxicology perspectives including cancer risk assessment, in silico, in vitro/in vigo testings, and regulatory aspects
  • 5. In silico/computational assessment for the evaluation of genotoxic impurities
  • 6.Preclinical assessment of genotoxic impurities an overview of current regulatroy guidance, available assays, and data interpretation
  • 7. Purification of lead compounds for early toxicology profiling sucs as ames and short-term non-GLP (good laboratory practice) toxicology tests
  • 8. Analysis of genotoxic impurities in pharmaceutical by gas chromatography-mass spectromatry
  • 9. Control of chloroethane in raw materials and drug substances using headspace/gas chromatograghy analysis
  • 10. Quantification of genotoxic impurities in active pharmaceutical ingredients
  • 11. Analytical testing and control for genotoxic impurities in drug substances
  • 12. Approaches to assess, analyze, and control genotoxic impurities in drug substance development
  • 13. Control and analysis of genotoxic impurities in drug substance development
  • 14. Salt formation of pharmaceutical compounds and associated genotoxic risks
  • 15. Identification and control of genotoxic degradation products
  • 16. Identifical and qualification of genotoxic impurities as leachables in drug products
  • 17. Pharmaceutical industry survey on genotoxic impurities and related topics