Textbook of drug design and discovery

Bibliographic Details
Other Authors: Krogsgaard-Larsen, Povl (Editor), Madsen, Ulf (Editor), Stromgaard, Kristian (Editor)
Format: Book
Language:English
Published: Florida : CRC Press c2017
Edition:5th ed
Subjects:
Table of Contents:
  • 1. Introduction to drug design and discovery
  • 2. Molecular recognition
  • 3. Ligand-based drug design
  • 4. Biostructure-based drug design
  • 5. Drug-like properties and decision making in medicinal chemistry
  • 6. Chemical biology
  • 7. Natural products in drug discovery
  • 8. In vivo imaging in drug discovery
  • 9. Peptide and protein drug design
  • 10. Prodrugs in drug design and development
  • 11. Enzyme inhibitors: biostructure-and mechanism-based design
  • 12. Receptors: structure, function, ?and pharmacology
  • 13. Ion channels: structure and function
  • 14. Neurotransmitter transporters: structure, function, and drug binding
  • 15. Gaba and glutamic acid receptor and transporter ligands