Synthesis and Evaluation of N-(3-Trifluoroacetylindol-
7-yl) Acetamides for Potential In Vitro Antiplasmodial Properties

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Synthesis and Evaluation of N-(3-Trifluoroacetylindol- 7-yl) Acetamides for Potential In Vitro Antiplasmodial Properties

A series of novel N-((2,5-diaryl-3-trifluoroacetyl)-1H-indol-7-yl)acetamides has been prepared via a successive and one-pot reaction sequence involving initial trifluoroacetic acid-mediated Beckmann rearrangement of the oximes derived from the 1-(2,5-diaryl-1H-indol-7-yl)ethanones, followed by tr...

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Bibliographic Details
Main Authors:	Malose J., Mphahlele, Mmakwena M., Mmonwa, Yee, Siew Choong
Format:	Article
Language:	English
Published:	MDPI 2017
Subjects:	R735-854 Medical education. Medical schools. Research
Online Access:	http://eprints.usm.my/37238/ http://eprints.usm.my/37238/1/%28Synthesis_and_Evaluation%29_molecules-22-01099.pdf

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