Antioxidative and photocytotoxic effects of standardized Clinacanthus nutans and Strobilanthes crispus extracts toward HepG2 liver cells

Introduction: The methanolic extracts of Clinacanthus nutans (CME) and Strobilanthes crispus (SME) are used in Malaysia as a complementary and alternative medicine for cancer. Objective: The present study aimed to determine the antioxidative and photocytotoxic effects of CME and SME toward liver...

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Main Authors: Tan, Sheri-Ann, Shi, Yun Lim, Chieu, Shie Law, Chen, Son Yue, Tze, Ven Poh, Saad, Wan Zuhainis, Ismail, Saila, Mohd Yusoff, Khatijah, Loke, Chui Fung
Format: Article
Language:English
Published: Medknow Publications and Media 2019
Online Access:http://psasir.upm.edu.my/id/eprint/80687/
http://psasir.upm.edu.my/id/eprint/80687/1/NUTAN.pdf
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author Tan, Sheri-Ann
Shi, Yun Lim
Chieu, Shie Law
Chen, Son Yue
Tze, Ven Poh
Saad, Wan Zuhainis
Ismail, Saila
Mohd Yusoff, Khatijah
Loke, Chui Fung
author_facet Tan, Sheri-Ann
Shi, Yun Lim
Chieu, Shie Law
Chen, Son Yue
Tze, Ven Poh
Saad, Wan Zuhainis
Ismail, Saila
Mohd Yusoff, Khatijah
Loke, Chui Fung
author_sort Tan, Sheri-Ann
building UPM Institutional Repository
collection Online Access
description Introduction: The methanolic extracts of Clinacanthus nutans (CME) and Strobilanthes crispus (SME) are used in Malaysia as a complementary and alternative medicine for cancer. Objective: The present study aimed to determine the antioxidative and photocytotoxic effects of CME and SME toward liver cancer cells. Materials and Methods: Cell‑based (2′,7′‑dichlorodihydrofluorescein diacetate) and chemical‑based (2,2‑diphenyl‑1‑picrylhydrazyl [DPPH]) experiments were utilized to determine the antioxidative properties of both herbal extracts. CME and SME were also tested for their photocytotoxic potentials after photodynamic therapy (PDT). Phytochemical analysis was performed to identify the phytocompounds present in the extracts. Results: Both the extracts demonstrated dose‑dependent DPPH radical scavenging activities, while SME was found to be a stronger reactive oxygen species scavenger than CME at all concentrations tested on liver cells. Interestingly, on PDT, HepG2 cells treated with SME and CME at nontoxic doses showed a decrease in cellular viability charting half‑maximal inhibitory concentration of 13.45 μg/mL and 81.03 μg/mL, respectively. Total phenolic content of SME (36.27 ± 1.31 mg GAE/g extract) was slightly higher than CME (31.76 ± 0.10 mg GAE/g extract). On the contrary, the total flavonoid content of CME (11.32 ± 0.28 mg QE/g extract) was approximately seven times more than SME (1.69 ± 0.03 mg QE/g extract). Phenolic acids, flavonoids, and pheophorbide‑a were identified in both extracts. In view of this, these phytocompounds present in CME and SME could lead to the observed beneficial effects. Conclusion: CME and SME, especially the latter, are strong antioxidants with photosensitizing potentials that should be further investigated.
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spelling upm-806872020-11-12T00:43:07Z http://psasir.upm.edu.my/id/eprint/80687/ Antioxidative and photocytotoxic effects of standardized Clinacanthus nutans and Strobilanthes crispus extracts toward HepG2 liver cells Tan, Sheri-Ann Shi, Yun Lim Chieu, Shie Law Chen, Son Yue Tze, Ven Poh Saad, Wan Zuhainis Ismail, Saila Mohd Yusoff, Khatijah Loke, Chui Fung Introduction: The methanolic extracts of Clinacanthus nutans (CME) and Strobilanthes crispus (SME) are used in Malaysia as a complementary and alternative medicine for cancer. Objective: The present study aimed to determine the antioxidative and photocytotoxic effects of CME and SME toward liver cancer cells. Materials and Methods: Cell‑based (2′,7′‑dichlorodihydrofluorescein diacetate) and chemical‑based (2,2‑diphenyl‑1‑picrylhydrazyl [DPPH]) experiments were utilized to determine the antioxidative properties of both herbal extracts. CME and SME were also tested for their photocytotoxic potentials after photodynamic therapy (PDT). Phytochemical analysis was performed to identify the phytocompounds present in the extracts. Results: Both the extracts demonstrated dose‑dependent DPPH radical scavenging activities, while SME was found to be a stronger reactive oxygen species scavenger than CME at all concentrations tested on liver cells. Interestingly, on PDT, HepG2 cells treated with SME and CME at nontoxic doses showed a decrease in cellular viability charting half‑maximal inhibitory concentration of 13.45 μg/mL and 81.03 μg/mL, respectively. Total phenolic content of SME (36.27 ± 1.31 mg GAE/g extract) was slightly higher than CME (31.76 ± 0.10 mg GAE/g extract). On the contrary, the total flavonoid content of CME (11.32 ± 0.28 mg QE/g extract) was approximately seven times more than SME (1.69 ± 0.03 mg QE/g extract). Phenolic acids, flavonoids, and pheophorbide‑a were identified in both extracts. In view of this, these phytocompounds present in CME and SME could lead to the observed beneficial effects. Conclusion: CME and SME, especially the latter, are strong antioxidants with photosensitizing potentials that should be further investigated. Medknow Publications and Media 2019 Article PeerReviewed text en http://psasir.upm.edu.my/id/eprint/80687/1/NUTAN.pdf Tan, Sheri-Ann and Shi, Yun Lim and Chieu, Shie Law and Chen, Son Yue and Tze, Ven Poh and Saad, Wan Zuhainis and Ismail, Saila and Mohd Yusoff, Khatijah and Loke, Chui Fung (2019) Antioxidative and photocytotoxic effects of standardized Clinacanthus nutans and Strobilanthes crispus extracts toward HepG2 liver cells. Pharmacognosy Magazine, 15 (65). pp. 613-620. ISSN 0973-1296; ESSN: 0976-4062 http://www.phcog.com/temp/PhcogMag1565613-105503_025550.pdf 10.4103/pm.pm_84_19
spellingShingle Tan, Sheri-Ann
Shi, Yun Lim
Chieu, Shie Law
Chen, Son Yue
Tze, Ven Poh
Saad, Wan Zuhainis
Ismail, Saila
Mohd Yusoff, Khatijah
Loke, Chui Fung
Antioxidative and photocytotoxic effects of standardized Clinacanthus nutans and Strobilanthes crispus extracts toward HepG2 liver cells
title Antioxidative and photocytotoxic effects of standardized Clinacanthus nutans and Strobilanthes crispus extracts toward HepG2 liver cells
title_full Antioxidative and photocytotoxic effects of standardized Clinacanthus nutans and Strobilanthes crispus extracts toward HepG2 liver cells
title_fullStr Antioxidative and photocytotoxic effects of standardized Clinacanthus nutans and Strobilanthes crispus extracts toward HepG2 liver cells
title_full_unstemmed Antioxidative and photocytotoxic effects of standardized Clinacanthus nutans and Strobilanthes crispus extracts toward HepG2 liver cells
title_short Antioxidative and photocytotoxic effects of standardized Clinacanthus nutans and Strobilanthes crispus extracts toward HepG2 liver cells
title_sort antioxidative and photocytotoxic effects of standardized clinacanthus nutans and strobilanthes crispus extracts toward hepg2 liver cells
url http://psasir.upm.edu.my/id/eprint/80687/
http://psasir.upm.edu.my/id/eprint/80687/
http://psasir.upm.edu.my/id/eprint/80687/
http://psasir.upm.edu.my/id/eprint/80687/1/NUTAN.pdf