Synthesis, in-vitro bioactivity evaluation and molecular docking of monosaccharide ester and fatty acid amide derivatives of 5-aminosalicylic acid

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Synthesis, in-vitro bioactivity evaluation and molecular docking of monosaccharide ester and fatty acid amide derivatives of 5-aminosalicylic acid

5-aminosalicylic acid (5-ASA), structurally related to the salicylates, is active in the treatment of inflammatory bowel disease (IBD). Since IBD is a high-incidence disease and considering that 5-ASA has been approved as one of the most effective and tolerable drug for the majority of patients in t...

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Bibliographic Details
Main Author:	Yousefi, Samira
Format:	Thesis
Language:	English
Published:	2016
Subjects:	Monosaccharides - Synthesis Salicylates - Therapeutic use
Online Access:	http://psasir.upm.edu.my/id/eprint/75446/ http://psasir.upm.edu.my/id/eprint/75446/1/FS%202016%208.pdf

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