Inhibition of hepatitis B virus assembly with synthetic peptides derived from the viral surface and core antigens

The long surface antigen (L-HBsAg) of hepatitis B virus (HBV) plays a central role in the production of infectious virions. During HBV morphogenesis, both the PreS and S domains of L-HBsAg form docking sites for the viral nucleocapsids. Thus, a compound that disrupts the interaction between the L-HB...

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Main Author: Tan, Wen Siang
Format: Article
Language:English
English
Published: Applied Microbiology, Molecular and Cellular Biosciences Research Foundation 2002
Online Access:http://psasir.upm.edu.my/id/eprint/34512/
http://psasir.upm.edu.my/id/eprint/34512/1/Inhibition%20of%20hepatitis%20B%20virus%20assembly%20with%20synthetic%20peptides%20derived%20from%20the%20viral%20surface%20and%20core%20antigens.pdf
http://psasir.upm.edu.my/id/eprint/34512/7/48_103.pdf
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author Tan, Wen Siang
author_facet Tan, Wen Siang
author_sort Tan, Wen Siang
building UPM Institutional Repository
collection Online Access
description The long surface antigen (L-HBsAg) of hepatitis B virus (HBV) plays a central role in the production of infectious virions. During HBV morphogenesis, both the PreS and S domains of L-HBsAg form docking sites for the viral nucleocapsids. Thus, a compound that disrupts the interaction between the L-HBsAg and nucleocapsids could serve as a therapeutic agent against the virus based upon inhibition of morphogenesis. Synthetic peptides correspond to the binding sites in L-HBsAg inhibited the association of L-HBsAg with core antigen (HBcAg). A synthetic peptide carrying the epitope for a monoclonal antibody to the PreS1 domain competed weakly with L-HBsAg for HBcAg, but peptides corresponding to a linear sequence at the tip of the nucleocapsid spike did not, showing that the competing peptide does not resemble the tip of the spike.
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institution Universiti Putra Malaysia
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language English
English
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publishDate 2002
publisher Applied Microbiology, Molecular and Cellular Biosciences Research Foundation
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spelling upm-345122024-08-08T01:32:16Z http://psasir.upm.edu.my/id/eprint/34512/ Inhibition of hepatitis B virus assembly with synthetic peptides derived from the viral surface and core antigens Tan, Wen Siang The long surface antigen (L-HBsAg) of hepatitis B virus (HBV) plays a central role in the production of infectious virions. During HBV morphogenesis, both the PreS and S domains of L-HBsAg form docking sites for the viral nucleocapsids. Thus, a compound that disrupts the interaction between the L-HBsAg and nucleocapsids could serve as a therapeutic agent against the virus based upon inhibition of morphogenesis. Synthetic peptides correspond to the binding sites in L-HBsAg inhibited the association of L-HBsAg with core antigen (HBcAg). A synthetic peptide carrying the epitope for a monoclonal antibody to the PreS1 domain competed weakly with L-HBsAg for HBcAg, but peptides corresponding to a linear sequence at the tip of the nucleocapsid spike did not, showing that the competing peptide does not resemble the tip of the spike. Applied Microbiology, Molecular and Cellular Biosciences Research Foundation 2002 Article PeerReviewed text en http://psasir.upm.edu.my/id/eprint/34512/1/Inhibition%20of%20hepatitis%20B%20virus%20assembly%20with%20synthetic%20peptides%20derived%20from%20the%20viral%20surface%20and%20core%20antigens.pdf text en http://psasir.upm.edu.my/id/eprint/34512/7/48_103.pdf Tan, Wen Siang (2002) Inhibition of hepatitis B virus assembly with synthetic peptides derived from the viral surface and core antigens. Journal of General and Applied Microbiology, 48 (2). pp. 103-107. ISSN 0022-1260; ESSN: 1349-8037 https://www.jstage.jst.go.jp/article/jgam/48/2/48_2_103/_article 10.2323/jgam.48.103
spellingShingle Tan, Wen Siang
Inhibition of hepatitis B virus assembly with synthetic peptides derived from the viral surface and core antigens
title Inhibition of hepatitis B virus assembly with synthetic peptides derived from the viral surface and core antigens
title_full Inhibition of hepatitis B virus assembly with synthetic peptides derived from the viral surface and core antigens
title_fullStr Inhibition of hepatitis B virus assembly with synthetic peptides derived from the viral surface and core antigens
title_full_unstemmed Inhibition of hepatitis B virus assembly with synthetic peptides derived from the viral surface and core antigens
title_short Inhibition of hepatitis B virus assembly with synthetic peptides derived from the viral surface and core antigens
title_sort inhibition of hepatitis b virus assembly with synthetic peptides derived from the viral surface and core antigens
url http://psasir.upm.edu.my/id/eprint/34512/
http://psasir.upm.edu.my/id/eprint/34512/
http://psasir.upm.edu.my/id/eprint/34512/
http://psasir.upm.edu.my/id/eprint/34512/1/Inhibition%20of%20hepatitis%20B%20virus%20assembly%20with%20synthetic%20peptides%20derived%20from%20the%20viral%20surface%20and%20core%20antigens.pdf
http://psasir.upm.edu.my/id/eprint/34512/7/48_103.pdf