Three new amides from Streptomyces sp. H7372

Three new amides, methyl phenatate A (1), actiphenamide (2) and actiphenol 1-β-D- glucopyranoside (3), along with thirteen known compounds, were isolated from the organic extract of a fermentation culture of Streptomyces sp. H7372. The structures were elucidated by spectroscopic methods including 1D...

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Main Authors: Cheenpracha, Sarot, Borris, Robert P., Tran, Tammy T., Jee, Jap Meng, Seow, Heng Fong, Cheah, Hwen Yee, Ho, Coy Choke, Chang, Leng Chee
Format: Article
Language:English
Published: Sociedade Brasileira de Química 2011
Online Access:http://psasir.upm.edu.my/id/eprint/24724/
http://psasir.upm.edu.my/id/eprint/24724/1/Three%20new%20amides%20from%20streptomyces%20sp.pdf
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author Cheenpracha, Sarot
Borris, Robert P.
Tran, Tammy T.
Jee, Jap Meng
Seow, Heng Fong
Cheah, Hwen Yee
Ho, Coy Choke
Chang, Leng Chee
author_facet Cheenpracha, Sarot
Borris, Robert P.
Tran, Tammy T.
Jee, Jap Meng
Seow, Heng Fong
Cheah, Hwen Yee
Ho, Coy Choke
Chang, Leng Chee
author_sort Cheenpracha, Sarot
building UPM Institutional Repository
collection Online Access
description Three new amides, methyl phenatate A (1), actiphenamide (2) and actiphenol 1-β-D- glucopyranoside (3), along with thirteen known compounds, were isolated from the organic extract of a fermentation culture of Streptomyces sp. H7372. The structures were elucidated by spectroscopic methods including 1D- and 2D-NMR techniques, and MS analyses. Cycloheximide (6) and cyclo(δAla-L- Val) (8) gave a clear zone of inhibition of Ras-Raf-1 interaction in the yeast two- hybrid assay which showed high potency with 10 and 25 mm clear ZOIs on SD His - and inactive on SD His + at 2.5 μg per disk, respectively.
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language English
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publishDate 2011
publisher Sociedade Brasileira de Química
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spelling upm-247242016-12-02T03:33:34Z http://psasir.upm.edu.my/id/eprint/24724/ Three new amides from Streptomyces sp. H7372 Cheenpracha, Sarot Borris, Robert P. Tran, Tammy T. Jee, Jap Meng Seow, Heng Fong Cheah, Hwen Yee Ho, Coy Choke Chang, Leng Chee Three new amides, methyl phenatate A (1), actiphenamide (2) and actiphenol 1-β-D- glucopyranoside (3), along with thirteen known compounds, were isolated from the organic extract of a fermentation culture of Streptomyces sp. H7372. The structures were elucidated by spectroscopic methods including 1D- and 2D-NMR techniques, and MS analyses. Cycloheximide (6) and cyclo(δAla-L- Val) (8) gave a clear zone of inhibition of Ras-Raf-1 interaction in the yeast two- hybrid assay which showed high potency with 10 and 25 mm clear ZOIs on SD His - and inactive on SD His + at 2.5 μg per disk, respectively. Sociedade Brasileira de Química 2011 Article PeerReviewed application/pdf en http://psasir.upm.edu.my/id/eprint/24724/1/Three%20new%20amides%20from%20streptomyces%20sp.pdf Cheenpracha, Sarot and Borris, Robert P. and Tran, Tammy T. and Jee, Jap Meng and Seow, Heng Fong and Cheah, Hwen Yee and Ho, Coy Choke and Chang, Leng Chee (2011) Three new amides from Streptomyces sp. H7372. Journal of the Brazilian Chemical Society, 22 (2). pp. 223-229. ISSN 0103-5053; ESSN: 1678-4790 10.1590/S0103-50532011000200006
spellingShingle Cheenpracha, Sarot
Borris, Robert P.
Tran, Tammy T.
Jee, Jap Meng
Seow, Heng Fong
Cheah, Hwen Yee
Ho, Coy Choke
Chang, Leng Chee
Three new amides from Streptomyces sp. H7372
title Three new amides from Streptomyces sp. H7372
title_full Three new amides from Streptomyces sp. H7372
title_fullStr Three new amides from Streptomyces sp. H7372
title_full_unstemmed Three new amides from Streptomyces sp. H7372
title_short Three new amides from Streptomyces sp. H7372
title_sort three new amides from streptomyces sp. h7372
url http://psasir.upm.edu.my/id/eprint/24724/
http://psasir.upm.edu.my/id/eprint/24724/
http://psasir.upm.edu.my/id/eprint/24724/1/Three%20new%20amides%20from%20streptomyces%20sp.pdf