Caspases-3 and -7 are activated in goniothalamin-induced apoptosis in human Jurkat T-cells

Goniothalamin, a plant styrylpyrone derivative isolated from Goniothalamus andersonii, induced apoptosis in Jurkat T-cells as assessed by the externalisation of phosphatidylserine. Immunoblotting showed processing of caspases-3 and -7 with the appearance of their catalytically active large subunits...

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Bibliographic Details
Main Authors: Inayat-Hussain, Salmaan H., Osman, Annuar B., Din, Laily B., Ali, Abdul M.
Format: Article
Language:English
Published: Federation of European Biochemical Societies 1999
Online Access:http://psasir.upm.edu.my/id/eprint/114448/
http://psasir.upm.edu.my/id/eprint/114448/1/114448.pdf
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Summary:Goniothalamin, a plant styrylpyrone derivative isolated from Goniothalamus andersonii, induced apoptosis in Jurkat T-cells as assessed by the externalisation of phosphatidylserine. Immunoblotting showed processing of caspases-3 and -7 with the appearance of their catalytically active large subunits of 17 and 19 kDa, respectively. Activation of these caspases was further evidenced by detection of poly(ADP-ribose) polymerase cleavage (PARP). Pre-treatment with the caspase inhibitor benzyloxycarbonyl-Val-Ala-Asp fluoromethyl ketone (Z-VAD.FMK) blocked apoptosis and the resultant cleavage of these caspases and PARP. Our results demonstrate that activation of at least two effector caspases is a key feature of goniothalamin-induced apoptosis in Jurkat T-cells.