Synthesis, characterization and molecular docking of hydroxyxanthone and renylated xanthone derivatives as potential aromatase inhibitor

QR Code

Synthesis, characterization and molecular docking of hydroxyxanthone and renylated xanthone derivatives as potential aromatase inhibitor

Xanthone is an important scaffold for the development of new drugs due to its various positions and types of attached substituents with specific functions. This makes xanthone and their derivatives capable of exhibiting a variety of cytotoxic and biological activities. By discovering new lead compou...

Full description

Bibliographic Details
Main Author:	Ramakrishnan, Shurutishria
Format:	Thesis
Language:	English English
Published:	2022
Subjects:	Xanthone Aromatase
Online Access:	http://psasir.upm.edu.my/id/eprint/112694/ http://psasir.upm.edu.my/id/eprint/112694/1/112694.pdf

Similar Items

One-pot two-component synthesis of halogenated xanthone, 3-o substituted xanthone, and prenylated xanthone derivatives as aromatase inhibitors
by: Ramakrishnan, Shurutishria, et al.
Published: (2023)

Extraction, physicochemical properties and antioxidant activities of xanthone from mangosteen (Garcinia mangostana Linn.) pericarp
by: Aboutorab, Nasrin
Published: (2017)

Extraction of xanthone derivatives from mangosteen (Garcinia mangostana L.) pericarp with virgin coconut oil by supercritical carbon dioxide
by: Kok, Siew Lee
Published: (2022)

Potent halogenated xanthone derivatives: synthesis, molecular docking and study on antityrosinase activity
by: Baharuddin, Fatin Farhana, et al.
Published: (2023)

Synthesis and molecular docking of carvone derivatives as a potential neuraminidase inhibitors
by: Jusoh, Noorakmar, et al.
Published: (2016)

Synthesis of thymidine phosphorylase inhibitor based on quinoxaline derivatives and their molecular docking study
by: Noor Barak, Almandil, et al.
Published: (2019)

Synthesis of thymidine phosphorylase inhibitor based on quinoxaline derivatives and their molecular docking study
by: Almandil, Noor Barak, et al.
Published: (2019)

Textured Renyl Entropy for Image Thresholding
by: Abu Shareha, Ahmad Adel, et al.
Published: (2008)

Double-blind randomized controlled trial of letrozole versus clomiphene citrate in subfertile women with polycystic ovarian syndrome
by: Amer, Saad A., et al.
Published: (2017)

Synthesis of new isoquinoline-base-oxadiazole derivatives as potent inhibitors of thymidine phosphorylase and molecular docking study
by: Zaman, Khalid, et al.
Published: (2019)

Xanthones and xanthone derivatives from Garcinia nitida
by: Ee, Gwendoline Cheng Lian, et al.
Published: (2007)

Synthesis, neuraminidase inhibition assay and molecular docking of carvone derivatives
by: Abd Hamid, Shafida
Published: (2019)

Evaluation of potential bacterial protease inhibitor properties of selected hydroxyquinoline derivatives : An in silico docking and molecular dynamics simulation approach
by: Riaz, Faiza, et al.
Published: (2023)

Leptin hormone changes in patients with poly cystic ovarian syndrome treated by aromatase inhibitors
by: Al Omari, Wafa, et al.
Published: (2018)

Improve product quantity of aromatase inhibitor from Nicotiana tabaccum by metabolic engineering techique
by: Amid, Azura, et al.
Published: (2010)

Molecular docking studies of selected medicinal drugs as dengue virus-2 protease inhibitors
by: Rufaidah Othman,, et al.
Published: (2017)

Synthesis And Molecular Docking Studies Of New Phenylisoxazole Quinoxaline-2-Amine Hybrids As Potential Α Amylase And Α-Glucosidase Inhibitors
by: Radzuan, Siti Nurshahira Mohd
Published: (2024)

Molecular docking of selected flavonoid compounds from nelumbo nucifera as potential pancreatic lipase inhibitor
by: Ghazali, Siti Nur Akmal, et al.
Published: (2017)

Computational quest for finding potential Ebola VP40 inhibitors: a molecular docking study
by: Mohamad Ariff Mohamad Yussoff,, et al.
Published: (2020)

A quest on finding new potential ebola vp40 inhibitors: molecular docking and molecular dynamics simulation studies
by: Mohamad Yussoff, Mohamad Ariff, et al.
Published: (2018)

Molecular docking analysis of curcumin analogues as human neutrophil elastase inhibitors
by: Narayanaswamy, Radhakrishnan, et al.
Published: (2014)

Molecular docking of substituted schiff bases derived from s-benzyldithiocarbazate as potential anticancer agents
by: How, Fiona Ni Foong
Published: (2018)

Synthesis of new anilinoquinazoline derivatives as potential anticancer agents: Antiproliferative activity, molecular docking and molecular dynamics studies / Muhammad Kumayl Abdul Wahab
by: Muhammad Kumayl , Abdul Wahab
Published: (2021)

Synthesis of benzylated amine-substituted xanthone derivatives and their antioxidant and anti-inflammatory activities
by: Wong, Ka Woong, et al.
Published: (2022)

Synthesis and investigation of anti-tyrosinase and antioxidant activity of new halogenated xanthone derivatives
by: Baharuddin, Fatin Farhana
Published: (2023)

Chemical synthesis of 1,3,8-trioxygenated xanthone derivatives and their cytotoxic activities
by: Tan, Su Chin
Published: (2011)

Synthesis and docking studies of 2,4,6-trihydroxy-3-geranylacetophenone analogs as potential lipoxygenase inhibitor
by: Chean, Hui Ng, et al.
Published: (2014)

Design, Synthesis, Molecular Docking And Cytotoxic Activity Of New Ortho-Hydroxy Chalcone And Pyrazoline Derivatives
by: Luhaibi, Maadh Jumaah Owaid
Published: (2019)

Synthesis, Cholinesterase Inhibitory Activity And Molecular Docking Study Of Piperidone-Grafted Pyrimidine And Thiazolopyrimidine Derivatives
by: Basiri, Alireza
Published: (2014)

Molecular docking unveils prospective inhibitors for the SARS-COV-2 main protease
by: Ahmad, Fawad, et al.
Published: (2021)

Molecular docking
by: Abduallah Alsafi, Hassen Mohammed, et al.
Published: (2011)

Synthesis, Characterisation And Molecular Docking Of Quinoxaline-isoxazole Hybrids As Potential Anti-hyperglycemic Agent
by: Phongphane, Lacksany
Published: (2024)

Synthesis and antioxidant activity of Prenylated Xanthones derived from 1,3,6-Trihydroxyxanthone.
by: Chan, Siew Ling
Published: (2013)

Synthesis, characterisation and cytotoxic activities of 1, 3, 6, 8 – tetraoxygenated xanthone derivatives
by: Lim, Shian Hoi
Published: (2011)

Development of diarylpentadienone analogues as alpha-glucosidase inhibitor: Synthesis, in vitro biological and in vivo toxicity evaluations, and molecular docking analysis
by: Maryam Aisyah, Abdullah, et al.
Published: (2020)

Cholinesterase inhibition activity and molecular docking study of eugenol derivatives
by: Khairunisa Mohd Zamli,, et al.
Published: (2021)

Cytotoxicity, antimutagenicity and molecular docking of benzimidazole derivatives as anticancer agents
by: Azahar, Nurul Hafizan
Published: (2021)

Synthesis and molecular docking of 2, 4, 5-trisubstituted-1,3-thiazole derivatives as antibacterial agents
by: Abdullah Ripain, Iswatun Hasanah, et al.
Published: (2018)

Elucidating the binding affinity of meso porphyrin derivatives with Bcl-2 through synthesis and molecular docking analysis
by: Yasothaa Ramaiyah,, et al.
Published: (2023)

Design, Synthesis and Molecular Docking Studies of Some Novel Spiro Derivatives By 1,3-Cycloaddition Reaction
by: Hasmaruddin, Nurul Syazana, et al.
Published: (2016)