Synthesis and Antibacterial Activity of Acetoxybenzoyl Thioureas with Aryl and Amino Acid Side Chains
A series of acetoxybenzoylthioureas derivatives with aryl and amino acid ester side chains were prepared by reaction of acetoxybenzoyl isothiocyanate, an acyloxy benzyl esterbased derivative of aspirin, with aryl amines or amino-functionalized amino acids with overall yields of 46–73%. The produc...
| Main Authors: | Zainab, Ngaini, Maya Asyikin, Mohd Ariff, Hasnain, Hussain, Er, Su Mei, Tang, Donna, Dyg Halimatulzahrah, Abang Kamaluddin |
|---|---|
| Format: | Article |
| Language: | English |
| Published: |
Taylor & Francis Group, LLC
2012
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| Subjects: | |
| Online Access: | http://ir.unimas.my/id/eprint/15578/ http://ir.unimas.my/id/eprint/15578/1/maya.pdf |
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