Synthesis of Glycosides Bearing Chalcone Derivatives via Ferrier Rearrangement

A series of glycoside derivatives bearing chalcones moieties has been synthesized. A convenient synthetic method was performed from the reaction of 3,4,6-tri-O-acetyl-D-glucal with (E)-1-(4-alkyloxyphenyl)-3-(4-hydroxy-phenyl)prop-2-en-1-one (2a-2c) employing OC rearrangement to afford C-glycoside...

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Main Authors: Zainab, Ngaini, Dayang H., Abang Kamaluddin
Format: Article
Language:English
Published: Institut Kimia Malaysia 2013
Subjects:
Online Access:http://ir.unimas.my/id/eprint/15569/
http://ir.unimas.my/id/eprint/15569/1/Synthesis%20of%20Glycosides%20Bearing%20Chalcone%20%28abstract%29.pdf
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author Zainab, Ngaini
Dayang H., Abang Kamaluddin
author_facet Zainab, Ngaini
Dayang H., Abang Kamaluddin
author_sort Zainab, Ngaini
building UNIMAS Institutional Repository
collection Online Access
description A series of glycoside derivatives bearing chalcones moieties has been synthesized. A convenient synthetic method was performed from the reaction of 3,4,6-tri-O-acetyl-D-glucal with (E)-1-(4-alkyloxyphenyl)-3-(4-hydroxy-phenyl)prop-2-en-1-one (2a-2c) employing OC rearrangement to afford C-glycoside 4a-c over prolonged reaction times, in the presence of BF3.OEt2 as a catalyst. The compounds differ in the length of alkyl groups, CnH2n+1, where n= 7, 8 and 9.
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spelling unimas-155692017-03-15T10:38:55Z http://ir.unimas.my/id/eprint/15569/ Synthesis of Glycosides Bearing Chalcone Derivatives via Ferrier Rearrangement Zainab, Ngaini Dayang H., Abang Kamaluddin QD Chemistry A series of glycoside derivatives bearing chalcones moieties has been synthesized. A convenient synthetic method was performed from the reaction of 3,4,6-tri-O-acetyl-D-glucal with (E)-1-(4-alkyloxyphenyl)-3-(4-hydroxy-phenyl)prop-2-en-1-one (2a-2c) employing OC rearrangement to afford C-glycoside 4a-c over prolonged reaction times, in the presence of BF3.OEt2 as a catalyst. The compounds differ in the length of alkyl groups, CnH2n+1, where n= 7, 8 and 9. Institut Kimia Malaysia 2013 Article PeerReviewed text en http://ir.unimas.my/id/eprint/15569/1/Synthesis%20of%20Glycosides%20Bearing%20Chalcone%20%28abstract%29.pdf Zainab, Ngaini and Dayang H., Abang Kamaluddin (2013) Synthesis of Glycosides Bearing Chalcone Derivatives via Ferrier Rearrangement. Malaysian Journal of Chemistry, 15 (1). 013-019. ISSN 1511-2292 https://www.researchgate.net/publication/291336464_Synthesis_of_Glycosides_Bearing_Chalcone_Derivatives_via_Ferrier_Rearrangement
spellingShingle QD Chemistry
Zainab, Ngaini
Dayang H., Abang Kamaluddin
Synthesis of Glycosides Bearing Chalcone Derivatives via Ferrier Rearrangement
title Synthesis of Glycosides Bearing Chalcone Derivatives via Ferrier Rearrangement
title_full Synthesis of Glycosides Bearing Chalcone Derivatives via Ferrier Rearrangement
title_fullStr Synthesis of Glycosides Bearing Chalcone Derivatives via Ferrier Rearrangement
title_full_unstemmed Synthesis of Glycosides Bearing Chalcone Derivatives via Ferrier Rearrangement
title_short Synthesis of Glycosides Bearing Chalcone Derivatives via Ferrier Rearrangement
title_sort synthesis of glycosides bearing chalcone derivatives via ferrier rearrangement
topic QD Chemistry
url http://ir.unimas.my/id/eprint/15569/
http://ir.unimas.my/id/eprint/15569/
http://ir.unimas.my/id/eprint/15569/1/Synthesis%20of%20Glycosides%20Bearing%20Chalcone%20%28abstract%29.pdf