Synthesis, molecular docking and tyrosinase inhibitory activity of the decorated methoxy sulfonamide chalcones : in vitro inhibitory effects and the possible binding mode
In this study, a series of sulfonamide chalcones derivatives was synthesized and its chemical structures were confirmed by spectral characteristics. The synthesized compounds were evaluated for their tyrosinase inhibitory activities along with molecular docking study. The tyrosinase inhibitory resul...
| Main Authors: | Thawanrat Kobkeatthawin, Suchada Chantrapromma, Thitipone Suwunwong, Lydia Rhyman, Choong, Yee Siew, Ponnadurai Ramasami |
|---|---|
| Format: | Article |
| Language: | English |
| Published: |
Penerbit Universiti Kebangsaan Malaysia
2021
|
| Online Access: | http://journalarticle.ukm.my/18058/ http://journalarticle.ukm.my/18058/1/9.pdf |
Similar Items
Bioactive compounds, antioxidant, xanthine oxidase inhibitory, tyrosinase inhibitory and anti-inflammatory activities of selected agro-industrial by-products
by: Oskoueian, Ehsan, et al.
Published: (2011)
by: Oskoueian, Ehsan, et al.
Published: (2011)
Antioxidant, cholinesterase and tyrosinase inhibitory activities of calophyllum symingtonianum and calophyllum depressinervosum
by: Aminudin, Nurul Iman, et al.
Published: (2015)
by: Aminudin, Nurul Iman, et al.
Published: (2015)
Antioxidant activity study and tyrosinase inhibitory study of Entada spiralis Ridl.
by: Syed Mohamad, Syarifah Nurul Akilah, et al.
Published: (2016)
by: Syed Mohamad, Syarifah Nurul Akilah, et al.
Published: (2016)
Antioxidant activity study and tyrosinase inhibitory screening of Entada spiralis Ridl. leaves
by: Syed Mohammad, Sharifah Nurul Akilah, et al.
Published: (2016)
by: Syed Mohammad, Sharifah Nurul Akilah, et al.
Published: (2016)
In vitro antioxidant, cholinesterase and tyrosinase inhibitory activities of calophyllum symingtonianum and calophyllum depressinervosum (guttiferae)
by: Aminudin, Nurul Iman, et al.
Published: (2015)
by: Aminudin, Nurul Iman, et al.
Published: (2015)
Phenolic composition, antioxidant, anti-wrinkles and tyrosinase inhibitory activities of cocoa pod extract
by: Abdul Karim, Azila, et al.
Published: (2014)
by: Abdul Karim, Azila, et al.
Published: (2014)
α-Glucosidase inhibitors: consistency of: in silico docking data with in vitro inhibitory data and inhibitory effect prediction of quercetin derivatives
by: Zhu, Jianzhong, et al.
Published: (2019)
by: Zhu, Jianzhong, et al.
Published: (2019)
Transformation of Melinjo seed micropowders into nanopowders enhances extractability of phenolic compounds and tyrosinase inhibitory activity
by: Vienna Saraswaty,, et al.
Published: (2019)
by: Vienna Saraswaty,, et al.
Published: (2019)
Tyrosinase inhibitory and antioxidant activities of
entada spiralis RIDL. (akar sintok) for the development of skin whitening product
by: Mat So'ad, Siti Zaiton, et al.
Published: (2017)
by: Mat So'ad, Siti Zaiton, et al.
Published: (2017)
Antioxidant, antimicrobial and tyrosinase inhibitory activities of xanthones isolated from artocarpus obtusus F.M. Jarrett
by: Mohd Hashim, Najihah, et al.
Published: (2012)
by: Mohd Hashim, Najihah, et al.
Published: (2012)
Evaluation Of Various Autodock
Molecular Docking Programmes In
Predicting The Neuraminidase
Inhibitory Activity
by: Raime, Nurul Nadia
Published: (2015)
by: Raime, Nurul Nadia
Published: (2015)
2-[(E)-2-(4-Ethoxyphenyl)ethenyl]-1-
methylquinolinium 4-fluorobenzenesulfonate
by: Hoong, Kun Fun, et al.
Published: (2014)
by: Hoong, Kun Fun, et al.
Published: (2014)
(E)-1-(2,4-Dinitrophenyl)-2-(3-ethoxy-4-hydroxybenzylidene)hydrazine
by: Fun, Hoong Kun, et al.
Published: (2014)
by: Fun, Hoong Kun, et al.
Published: (2014)
(E)-4-Methoxy-N00-(2,4,5-trimethoxybenzylidene)
benzohydrazide hemihydrate
by: Chantrapromma, Suchada, et al.
Published: (2014)
by: Chantrapromma, Suchada, et al.
Published: (2014)
Design and Synthesis of Chalcone Derivatives as Potent Tyrosinase Inhibitors and Their Structural Activity Relationship
by: Akhtar, Muhammad Nadeem, et al.
Published: (2015)
by: Akhtar, Muhammad Nadeem, et al.
Published: (2015)
Synthesis, Cholinesterase Inhibitory Activity And Molecular Docking Study Of Piperidone-Grafted Pyrimidine And Thiazolopyrimidine Derivatives
by: Basiri, Alireza
Published: (2014)
by: Basiri, Alireza
Published: (2014)
Anti–elastase, anti–tyrosinase and matrix metalloproteinase–1 inhibitory activity of earthworm extracts as potential new anti–aging agent
by: Azmi, Nurhazirah, et al.
Published: (2014)
by: Azmi, Nurhazirah, et al.
Published: (2014)
Nanocrystalline cellulose decorated quantum dots based tyrosinase biosensor for phenol determination
by: Abd Manan, Fariza Aina, et al.
Published: (2019)
by: Abd Manan, Fariza Aina, et al.
Published: (2019)
Bis{2-methoxy-6-[(E)-(4-methylbenzyl)-iminomethyl]phenolato}palladium(II) chloroform monosolvate
by: Bahron, Hadariah, et al.
Published: (2014)
by: Bahron, Hadariah, et al.
Published: (2014)
Inhibitory activity of cyclohexenyl chalcone derivatives and flavonoids of fingerroot, Boesenbergia rotunda (L.), towards dengue-2 virus NS3 protease.
by: Tan, Siew Kiat *, et al.
Published: (2006)
by: Tan, Siew Kiat *, et al.
Published: (2006)
Investigation of α‐glucosidase inhibitory metabolites from Tetracera scandens leaves by GC–MS metabolite profiling and docking studies
by: Ahmed, Nokhala, et al.
Published: (2020)
by: Ahmed, Nokhala, et al.
Published: (2020)
Investigation of α-glucosidase inhibitory metabolites from Tetracera scandens leaves by GC–MS metabolite profiling and docking studies
by: Nokhala, Ahmed, et al.
Published: (2020)
by: Nokhala, Ahmed, et al.
Published: (2020)
Biosensor based on tyrosinase immobilized on graphene decorated gold nanoparticle/chitosan for phenolic detection in aqueous
by: Mohamed Fartas, Fuzi, et al.
Published: (2017)
by: Mohamed Fartas, Fuzi, et al.
Published: (2017)
The role of inhibitory control in task switching
by: Yang, Violet Hye-Won
Published: (2010)
by: Yang, Violet Hye-Won
Published: (2010)
Handedness and the excitability of cortical inhibitory circuits
by: Reid, Campbell S., et al.
Published: (2012)
by: Reid, Campbell S., et al.
Published: (2012)
Synthesis, Cytotoxicity Study, And Molecular Docking Of New Imidazole-Based Chalcone And Pyrazoline Hybrids
by: Bakar, Bazri Izwan
Published: (2023)
by: Bakar, Bazri Izwan
Published: (2023)
Overexpression of host furin protease and inhibitory activities of synthetic chalcones- and azepines- derivative compounds toward dengue virus type-2 / Khuzaidatul Azidah Ahmad Nazri
by: Ahmad Nazri, Khuzaidatul Azidah
Published: (2016)
by: Ahmad Nazri, Khuzaidatul Azidah
Published: (2016)
Inhibitory effects of Manihot esculenta extracts on food-borne pathogens and their antioxidant properties: supercritical fluid extraction, statistical analysis, and molecular docking study
by: Ahmad, Mohammad Norazmi, et al.
Published: (2020)
by: Ahmad, Mohammad Norazmi, et al.
Published: (2020)
Individual differences in anxiety in relation to
inhibitory processes
by: Thurston, Meghan Dory
Published: (2011)
by: Thurston, Meghan Dory
Published: (2011)
Ubiquitous occurrence of sulfonamides in tropical Asian waters.
by: Shimizu, Akiko, et al.
Published: (2013)
by: Shimizu, Akiko, et al.
Published: (2013)
Minimum Inhibitory Concentration (MIC) and the Non-Inhibitory Concentration (NIC) values of Salvia officinalis methanolic extract against Aeromonas hydrophila
by: Ismail, Ahmad Syazwan, et al.
Published: (2022)
by: Ismail, Ahmad Syazwan, et al.
Published: (2022)
A computational docking analysis of chalcone synthase receptor and substrates in Boesenbergia rotunda / Ragaventhan Sanmugavelan
by: Ragaventhan , Sanmugavelan
Published: (2019)
by: Ragaventhan , Sanmugavelan
Published: (2019)
Design, Synthesis, Molecular
Docking And Cytotoxic Activity Of
New Ortho-Hydroxy Chalcone And
Pyrazoline Derivatives
by: Luhaibi, Maadh Jumaah Owaid
Published: (2019)
by: Luhaibi, Maadh Jumaah Owaid
Published: (2019)
Electrochemical tyrosinase biosensor based on cellulose nanocrystals decorated with CdS quantum dots and Fe₃O₄ nanoparticles for determination of phenol
by: Abd Manan, Fariza Aina
Published: (2018)
by: Abd Manan, Fariza Aina
Published: (2018)
2-acetylthiophene thiosemicarbazone as mushroom tyrosinase inhibitor: insights from kinetic, RDG, molecular docking, and DFT studies
by: Ahmad, Mohammad Norazmi, et al.
Published: (2019)
by: Ahmad, Mohammad Norazmi, et al.
Published: (2019)
Cannabinoid CB1 receptor binding and acetylcholinesterase
inhibitory activity of Sceletium tortuosum L.
by: Lubbe, A., et al.
Published: (2010)
by: Lubbe, A., et al.
Published: (2010)
Cannabinoid CB1 receptor binding and acetylcholinesterase
inhibitory activity of Sceletium tortuosum L.
by: Lubbe, Andrea, et al.
Published: (2010)
by: Lubbe, Andrea, et al.
Published: (2010)
Inhibitory effects of compounds from Zingiberaceae species on platelet activating factor receptor binding
by: Jantan, Ibrahim, et al.
Published: (2004)
by: Jantan, Ibrahim, et al.
Published: (2004)
α-Glucosidase inhibitory activity of selected Malaysian plants
by: Mohd Bukhari, Dzatil Awanis, et al.
Published: (2017)
by: Mohd Bukhari, Dzatil Awanis, et al.
Published: (2017)
Pancreatic lipase inhibitory potential of selected Malaysian plants
by: Alias, Norsyuhada, et al.
Published: (2014)
by: Alias, Norsyuhada, et al.
Published: (2014)
Similar Items
-
Bioactive compounds, antioxidant, xanthine oxidase inhibitory, tyrosinase inhibitory and anti-inflammatory activities of selected agro-industrial by-products
by: Oskoueian, Ehsan, et al.
Published: (2011) -
Antioxidant, cholinesterase and tyrosinase inhibitory activities of calophyllum symingtonianum and calophyllum depressinervosum
by: Aminudin, Nurul Iman, et al.
Published: (2015) -
Antioxidant activity study and tyrosinase inhibitory study of Entada spiralis Ridl.
by: Syed Mohamad, Syarifah Nurul Akilah, et al.
Published: (2016) -
Antioxidant activity study and tyrosinase inhibitory screening of Entada spiralis Ridl. leaves
by: Syed Mohammad, Sharifah Nurul Akilah, et al.
Published: (2016) -
In vitro antioxidant, cholinesterase and tyrosinase inhibitory activities of calophyllum symingtonianum and calophyllum depressinervosum (guttiferae)
by: Aminudin, Nurul Iman, et al.
Published: (2015)