Total syntheses of shizukaols A and E

Shizukaols possess a common heptacyclic framework containing more than ten contiguousstereocenters and potential biological activities. Here we report that the total syntheses ofshizukaols A (1)and E(2), two lindenane-type dimers from the Chloranthaceae family, areachieved via a modified biomimetic...

Full description

Bibliographic Details
Main Authors: Wu, Jian-Li, Lu, Yin-Suo, Tang, Bencan, Peng, Xiao-Shui
Format: Article
Language:English
Published: Springer Nature Publishing 2018
Online Access:https://eprints.nottingham.ac.uk/56370/
_version_ 1848799319215308800
author Wu, Jian-Li
Lu, Yin-Suo
Tang, Bencan
Peng, Xiao-Shui
author_facet Wu, Jian-Li
Lu, Yin-Suo
Tang, Bencan
Peng, Xiao-Shui
author_sort Wu, Jian-Li
building Nottingham Research Data Repository
collection Online Access
description Shizukaols possess a common heptacyclic framework containing more than ten contiguousstereocenters and potential biological activities. Here we report that the total syntheses ofshizukaols A (1)and E(2), two lindenane-type dimers from the Chloranthaceae family, areachieved via a modified biomimetic Diels–Alder reaction. The common crucial biomimetic diene23and ethylene species (6,17) are obtained through either a highlyZ-selective olefination ofα-siloxy ketone with ynolate anions or an intramolecular Horner–Wadsworth–Emmons olefinationfrom commercially available Wieland–Miescher ketone (7). This synthetic approach here opensup practical avenues for the total syntheses of the intriguing Chloranthaceae family members, aswell as the understanding of their relevant biological action in nature
first_indexed 2025-11-14T20:33:46Z
format Article
id nottingham-56370
institution University of Nottingham Malaysia Campus
institution_category Local University
language English
last_indexed 2025-11-14T20:33:46Z
publishDate 2018
publisher Springer Nature Publishing
recordtype eprints
repository_type Digital Repository
spelling nottingham-563702019-03-27T16:51:19Z https://eprints.nottingham.ac.uk/56370/ Total syntheses of shizukaols A and E Wu, Jian-Li Lu, Yin-Suo Tang, Bencan Peng, Xiao-Shui Shizukaols possess a common heptacyclic framework containing more than ten contiguousstereocenters and potential biological activities. Here we report that the total syntheses ofshizukaols A (1)and E(2), two lindenane-type dimers from the Chloranthaceae family, areachieved via a modified biomimetic Diels–Alder reaction. The common crucial biomimetic diene23and ethylene species (6,17) are obtained through either a highlyZ-selective olefination ofα-siloxy ketone with ynolate anions or an intramolecular Horner–Wadsworth–Emmons olefinationfrom commercially available Wieland–Miescher ketone (7). This synthetic approach here opensup practical avenues for the total syntheses of the intriguing Chloranthaceae family members, aswell as the understanding of their relevant biological action in nature Springer Nature Publishing 2018-10-02 Article PeerReviewed application/pdf en cc_by https://eprints.nottingham.ac.uk/56370/7/s41467-018-06245-7.pdf Wu, Jian-Li, Lu, Yin-Suo, Tang, Bencan and Peng, Xiao-Shui (2018) Total syntheses of shizukaols A and E. Nature Communications, 9 . 4040/1-4040/7. ISSN 2041-1723 http://dx.doi.org/10.1038/s41467-018-06245-7 doi:10.1038/s41467-018-06245-7 doi:10.1038/s41467-018-06245-7
spellingShingle Wu, Jian-Li
Lu, Yin-Suo
Tang, Bencan
Peng, Xiao-Shui
Total syntheses of shizukaols A and E
title Total syntheses of shizukaols A and E
title_full Total syntheses of shizukaols A and E
title_fullStr Total syntheses of shizukaols A and E
title_full_unstemmed Total syntheses of shizukaols A and E
title_short Total syntheses of shizukaols A and E
title_sort total syntheses of shizukaols a and e
url https://eprints.nottingham.ac.uk/56370/
https://eprints.nottingham.ac.uk/56370/
https://eprints.nottingham.ac.uk/56370/