Expedient synthesis of an atypical oxazolidinone compound library

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Expedient synthesis of an atypical oxazolidinone compound library

In order to address the current downturn in the drug discovery pipeline, initiatives are being undertaken to synthesise screening libraries of sp3-rich, low molecular weight compounds. As part of the European Lead Factory initiative, the synthesis and derivatisation of a simple hexahydrooxazolo[5,4-...

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Bibliographic Details
Main Authors:	Cully, Sarah J., Storr, Thomas E., Rawling, Michael J., Abeysena, Induka R., Hamza, Daniel, Jones, Geraint, Pearce, Christopher A., Quddus, Abdul, Lewis, William, Stockmand, Robert A.
Format:	Article
Published:	Elsevier 2016
Subjects:	sp3-rich; Library; Bicyclic; Scaffold; Oxazolidinone
Online Access:	https://eprints.nottingham.ac.uk/42754/

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