The design, synthesis and characterisation of subtype selective dipeptide-linked fluorescent ligands for human β1 and β2–adrenoceptors

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The design, synthesis and characterisation of subtype selective dipeptide-linked fluorescent ligands for human β1 and β2–adrenoceptors

Beta-adrenoceptors belong to the superfamily of G-protein coupled receptors (GPCR) and remain an important target for drug discovery. The complexity of GPCR pharmacology in terms of its signaling profile has led to a desire to further the study of receptor-ligand interaction and obtain more detaile...

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Bibliographic Details
Main Author:	Santu, L.T.
Format:	Thesis (University of Nottingham only)
Language:	English
Published:	2017
Subjects:	Fluorescent ligands Beta adrenoceptors binding asays
Online Access:	https://eprints.nottingham.ac.uk/40085/

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