Synthesis of triazole-linked morpholino oligonucleotides via Cu1 catalysed cycloaddition

Triazole-linked morpholino (TLMO) oligonucleic acids were synthesised using the CuI catalysed (3 + 2) azide–alkyne cycloaddition (CuAAC) reaction. The modified DNA analogues were incorporated into 13-mer sequences via solid phase synthesis. UV melting experiments showed that the TLMO modification gi...

Full description

Bibliographic Details
Main Authors: Palframan, Matthew J., Alharthy, Rima D., Powalowska, Paulina K., Hayes, Christopher J.
Format: Article
Published: Royal Society of Chemistry 2016
Online Access:https://eprints.nottingham.ac.uk/35070/
_version_ 1848794996685144064
author Palframan, Matthew J.
Alharthy, Rima D.
Powalowska, Paulina K.
Hayes, Christopher J.
author_facet Palframan, Matthew J.
Alharthy, Rima D.
Powalowska, Paulina K.
Hayes, Christopher J.
author_sort Palframan, Matthew J.
building Nottingham Research Data Repository
collection Online Access
description Triazole-linked morpholino (TLMO) oligonucleic acids were synthesised using the CuI catalysed (3 + 2) azide–alkyne cycloaddition (CuAAC) reaction. The modified DNA analogues were incorporated into 13-mer sequences via solid phase synthesis. UV melting experiments showed that the TLMO modification gives higher Tm values than the corresponding TLDNA modification.
first_indexed 2025-11-14T19:25:04Z
format Article
id nottingham-35070
institution University of Nottingham Malaysia Campus
institution_category Local University
last_indexed 2025-11-14T19:25:04Z
publishDate 2016
publisher Royal Society of Chemistry
recordtype eprints
repository_type Digital Repository
spelling nottingham-350702020-05-04T17:36:55Z https://eprints.nottingham.ac.uk/35070/ Synthesis of triazole-linked morpholino oligonucleotides via Cu1 catalysed cycloaddition Palframan, Matthew J. Alharthy, Rima D. Powalowska, Paulina K. Hayes, Christopher J. Triazole-linked morpholino (TLMO) oligonucleic acids were synthesised using the CuI catalysed (3 + 2) azide–alkyne cycloaddition (CuAAC) reaction. The modified DNA analogues were incorporated into 13-mer sequences via solid phase synthesis. UV melting experiments showed that the TLMO modification gives higher Tm values than the corresponding TLDNA modification. Royal Society of Chemistry 2016-02-16 Article PeerReviewed Palframan, Matthew J., Alharthy, Rima D., Powalowska, Paulina K. and Hayes, Christopher J. (2016) Synthesis of triazole-linked morpholino oligonucleotides via Cu1 catalysed cycloaddition. Organic and Biomolecular Chemistry, 14 . pp. 3112-3119. ISSN 1477-0520 http://dx.doi.org/10.1039/C6OB00007J 10.1039/C6OB00007J 10.1039/C6OB00007J 10.1039/C6OB00007J
spellingShingle Palframan, Matthew J.
Alharthy, Rima D.
Powalowska, Paulina K.
Hayes, Christopher J.
Synthesis of triazole-linked morpholino oligonucleotides via Cu1 catalysed cycloaddition
title Synthesis of triazole-linked morpholino oligonucleotides via Cu1 catalysed cycloaddition
title_full Synthesis of triazole-linked morpholino oligonucleotides via Cu1 catalysed cycloaddition
title_fullStr Synthesis of triazole-linked morpholino oligonucleotides via Cu1 catalysed cycloaddition
title_full_unstemmed Synthesis of triazole-linked morpholino oligonucleotides via Cu1 catalysed cycloaddition
title_short Synthesis of triazole-linked morpholino oligonucleotides via Cu1 catalysed cycloaddition
title_sort synthesis of triazole-linked morpholino oligonucleotides via cu1 catalysed cycloaddition
url https://eprints.nottingham.ac.uk/35070/
https://eprints.nottingham.ac.uk/35070/
https://eprints.nottingham.ac.uk/35070/