Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines
Cu-catalyzed three-component couplings of vinylazaarenes, B2(pin)2, and N-Boc imines are described. Oxidation of the initially formed boronate gives azaarene-containing, Boc-protected amino alcohols with reasonable to good diastereoselectivities.
| Main Authors: | , , |
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| Format: | Article |
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Royal Society of Chemistry
2016
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| Online Access: | https://eprints.nottingham.ac.uk/31806/ |
| _version_ | 1848794275914973184 |
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| author | Smith, Joshua J. Best, Daniel Lam, Hon Wai |
| author_facet | Smith, Joshua J. Best, Daniel Lam, Hon Wai |
| author_sort | Smith, Joshua J. |
| building | Nottingham Research Data Repository |
| collection | Online Access |
| description | Cu-catalyzed three-component couplings of vinylazaarenes, B2(pin)2, and N-Boc imines are described. Oxidation of the initially formed boronate gives azaarene-containing, Boc-protected amino alcohols with reasonable to good diastereoselectivities. |
| first_indexed | 2025-11-14T19:13:37Z |
| format | Article |
| id | nottingham-31806 |
| institution | University of Nottingham Malaysia Campus |
| institution_category | Local University |
| last_indexed | 2025-11-14T19:13:37Z |
| publishDate | 2016 |
| publisher | Royal Society of Chemistry |
| recordtype | eprints |
| repository_type | Digital Repository |
| spelling | nottingham-318062020-05-04T17:36:50Z https://eprints.nottingham.ac.uk/31806/ Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines Smith, Joshua J. Best, Daniel Lam, Hon Wai Cu-catalyzed three-component couplings of vinylazaarenes, B2(pin)2, and N-Boc imines are described. Oxidation of the initially formed boronate gives azaarene-containing, Boc-protected amino alcohols with reasonable to good diastereoselectivities. Royal Society of Chemistry 2016-02-17 Article PeerReviewed Smith, Joshua J., Best, Daniel and Lam, Hon Wai (2016) Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines. Chemical Communications . ISSN 1364-548X http://pubs.rsc.org/en/Content/ArticleLanding/2016/CC/C6CC00603E#!divAbstract doi:10.1039/C6CC00603E doi:10.1039/C6CC00603E |
| spellingShingle | Smith, Joshua J. Best, Daniel Lam, Hon Wai Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines |
| title | Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines |
| title_full | Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines |
| title_fullStr | Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines |
| title_full_unstemmed | Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines |
| title_short | Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines |
| title_sort | copper-catalyzed borylative coupling of vinylazaarenes and n-boc imines |
| url | https://eprints.nottingham.ac.uk/31806/ https://eprints.nottingham.ac.uk/31806/ https://eprints.nottingham.ac.uk/31806/ |