A glycopeptide dendrimer inhibitor of the galactose specific lectin LecA & of Pseudomonas aeruginosa biofilms

Biofilm inhibition is achieved with a phenylgalactosyl peptide dendrimer (see picture) that binds to the galactose-specific lectin LecA of P. aeruginosa. The multivalency of the ligands is critical for biofilm inhibition, although the nature of the linker between the peptide dendrimer and the galact...

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Main Authors: Kadam, Rameshwar U., Bergmann, Myriam, Hurley, Matthew, Garg, Divita, Cacciarini, Martina, Swiderska, Magdalena A., Nativi, Cristina, Sattler, Michael, Smyth, Alan R., Williams, Paul, Cámara, Miguel, Stocker, Achim, Darbre, Tamis, Reymond, Jean-Louis
Format: Article
Published: Wiley-VCH Verlag 2011
Online Access:https://eprints.nottingham.ac.uk/2843/
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author Kadam, Rameshwar U.
Bergmann, Myriam
Hurley, Matthew
Garg, Divita
Cacciarini, Martina
Swiderska, Magdalena A.
Nativi, Cristina
Sattler, Michael
Smyth, Alan R.
Williams, Paul
Cámara, Miguel
Stocker, Achim
Darbre, Tamis
Reymond, Jean-Louis
author_facet Kadam, Rameshwar U.
Bergmann, Myriam
Hurley, Matthew
Garg, Divita
Cacciarini, Martina
Swiderska, Magdalena A.
Nativi, Cristina
Sattler, Michael
Smyth, Alan R.
Williams, Paul
Cámara, Miguel
Stocker, Achim
Darbre, Tamis
Reymond, Jean-Louis
author_sort Kadam, Rameshwar U.
building Nottingham Research Data Repository
collection Online Access
description Biofilm inhibition is achieved with a phenylgalactosyl peptide dendrimer (see picture) that binds to the galactose-specific lectin LecA of P. aeruginosa. The multivalency of the ligands is critical for biofilm inhibition, although the nature of the linker between the peptide dendrimer and the galactose can provide additional contacts to the lectin and also has an effect on the interaction.
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institution University of Nottingham Malaysia Campus
institution_category Local University
last_indexed 2025-11-14T18:19:48Z
publishDate 2011
publisher Wiley-VCH Verlag
recordtype eprints
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spelling nottingham-28432020-05-04T16:31:42Z https://eprints.nottingham.ac.uk/2843/ A glycopeptide dendrimer inhibitor of the galactose specific lectin LecA & of Pseudomonas aeruginosa biofilms Kadam, Rameshwar U. Bergmann, Myriam Hurley, Matthew Garg, Divita Cacciarini, Martina Swiderska, Magdalena A. Nativi, Cristina Sattler, Michael Smyth, Alan R. Williams, Paul Cámara, Miguel Stocker, Achim Darbre, Tamis Reymond, Jean-Louis Biofilm inhibition is achieved with a phenylgalactosyl peptide dendrimer (see picture) that binds to the galactose-specific lectin LecA of P. aeruginosa. The multivalency of the ligands is critical for biofilm inhibition, although the nature of the linker between the peptide dendrimer and the galactose can provide additional contacts to the lectin and also has an effect on the interaction. Wiley-VCH Verlag 2011-11-04 Article PeerReviewed Kadam, Rameshwar U., Bergmann, Myriam, Hurley, Matthew, Garg, Divita, Cacciarini, Martina, Swiderska, Magdalena A., Nativi, Cristina, Sattler, Michael, Smyth, Alan R., Williams, Paul, Cámara, Miguel, Stocker, Achim, Darbre, Tamis and Reymond, Jean-Louis (2011) A glycopeptide dendrimer inhibitor of the galactose specific lectin LecA & of Pseudomonas aeruginosa biofilms. Angewandte Chemie International Edition, 50 (45). pp. 10631-10635. ISSN 1433-7851 http://onlinelibrary.wiley.com/doi/10.1002/anie.201104342/abstract doi:10.1002/anie.201104342 doi:10.1002/anie.201104342
spellingShingle Kadam, Rameshwar U.
Bergmann, Myriam
Hurley, Matthew
Garg, Divita
Cacciarini, Martina
Swiderska, Magdalena A.
Nativi, Cristina
Sattler, Michael
Smyth, Alan R.
Williams, Paul
Cámara, Miguel
Stocker, Achim
Darbre, Tamis
Reymond, Jean-Louis
A glycopeptide dendrimer inhibitor of the galactose specific lectin LecA & of Pseudomonas aeruginosa biofilms
title A glycopeptide dendrimer inhibitor of the galactose specific lectin LecA & of Pseudomonas aeruginosa biofilms
title_full A glycopeptide dendrimer inhibitor of the galactose specific lectin LecA & of Pseudomonas aeruginosa biofilms
title_fullStr A glycopeptide dendrimer inhibitor of the galactose specific lectin LecA & of Pseudomonas aeruginosa biofilms
title_full_unstemmed A glycopeptide dendrimer inhibitor of the galactose specific lectin LecA & of Pseudomonas aeruginosa biofilms
title_short A glycopeptide dendrimer inhibitor of the galactose specific lectin LecA & of Pseudomonas aeruginosa biofilms
title_sort glycopeptide dendrimer inhibitor of the galactose specific lectin leca & of pseudomonas aeruginosa biofilms
url https://eprints.nottingham.ac.uk/2843/
https://eprints.nottingham.ac.uk/2843/
https://eprints.nottingham.ac.uk/2843/