Synthesis and molecular docking of 2, 4, 5-trisubstituted-1,3-thiazole derivatives as antibacterial agents
The emergence of antibiotic resistance against bacterial strains has attracted great interest in the discovery and development of new antibacterial agents. Thiazole derivatives have been widely used in the biological as well as pharmacological fields and their efficiency as pharmaceutical drugs are...
| Main Authors: | Abdullah Ripain, Iswatun Hasanah, Roslan, Norashikin, Norshahimi, Nurul Shazana, Mohamed Salleh, Siti Salwa, Muhamad Bunnori, Noraslinda, Ngah, Nurziana |
|---|---|
| Format: | Proceeding Paper |
| Language: | English English |
| Published: |
2018
|
| Subjects: | |
| Online Access: | http://irep.iium.edu.my/67300/ http://irep.iium.edu.my/67300/1/SKAM_Poster.pdf http://irep.iium.edu.my/67300/7/67300%20SYNTHESIS%20AND%20MOLECULAR%20DOCKING.pdf |
Similar Items
Synthesis and molecular docking of 2,4,5-trisubstituted- 1,3-thiazole derivatives as antibacterial agents = Sintesis dan penyatuan molekul terbitan 1,3-tiazol berpenggantian-2,4,5 sebagai agen antibakteria
by: Abdullah Ripain, Iswatun Hasanah, et al.
Published: (2019)
by: Abdullah Ripain, Iswatun Hasanah, et al.
Published: (2019)
New 2,4,5-trisubstituted-1,3-thiazole derivatives: synthesis, in vitro antimicrobial activity and in silico study
by: Abdullah Ripain, Iswatun Hasanah, et al.
Published: (2020)
by: Abdullah Ripain, Iswatun Hasanah, et al.
Published: (2020)
Design, synthesis and characterization of 2,4-disubstituted-1,3 thiazole amino acid derivatives towards its applications on antimicrobial and antioxidant activities
by: Ngah, Nurziana, et al.
Published: (2018)
by: Ngah, Nurziana, et al.
Published: (2018)
Wound Healing Activity of Pyrazole-thiazole Derivatives of Curcumin Through the Docking, Pharmacokinetics, MD Simulation and MM/GBSA Approaches
by: Forid, Md Shaekh, et al.
Published: (2024)
by: Forid, Md Shaekh, et al.
Published: (2024)
Synthesis and molecular docking of carvone derivatives as a potential neuraminidase inhibitors
by: Jusoh, Noorakmar, et al.
Published: (2016)
by: Jusoh, Noorakmar, et al.
Published: (2016)
One-pot synthesis of thiazole hydrazones in water
by: Tan, Kit Lin
Published: (2018)
by: Tan, Kit Lin
Published: (2018)
Design and synthesis of indole-thiazole based inhibitors of UDP-galactopyranose mutase
by: Tie, Ding Yee
Published: (2013)
by: Tie, Ding Yee
Published: (2013)
Revealing the potency of 1,3,5-trisubstituted pyrazoline as antimalaria through combination of in silico studies
by: Rasyid, Herlina, et al.
Published: (2023)
by: Rasyid, Herlina, et al.
Published: (2023)
Synthesis, Characterization And
Microbial Activity Of New Thiazole,
Thiazolidinone, Thiadiazole And
Phenylacrylohydrazide Substituted
Coumarin Derivatives
by: Yusuf Zai, Samina Khan
Published: (2015)
by: Yusuf Zai, Samina Khan
Published: (2015)
Cytotoxicity, antimutagenicity and molecular docking of benzimidazole derivatives as anticancer agents
by: Azahar, Nurul Hafizan
Published: (2021)
by: Azahar, Nurul Hafizan
Published: (2021)
Synthesis, in-vitro and in silico studies of azo-based calix[4]arenes as antibacterial agent and neuraminidase inhibitor: a new look into an old scaffold
by: Ali, Yousaf, et al.
Published: (2018)
by: Ali, Yousaf, et al.
Published: (2018)
Molecular docking of substituted schiff bases derived from s-benzyldithiocarbazate as potential anticancer agents
by: How, Fiona Ni Foong
Published: (2018)
by: How, Fiona Ni Foong
Published: (2018)
Design, Synthesis and Molecular Docking Studies of Some Novel Spiro Derivatives By 1,3-Cycloaddition Reaction
by: Hasmaruddin, Nurul Syazana, et al.
Published: (2016)
by: Hasmaruddin, Nurul Syazana, et al.
Published: (2016)
Chemical and antibacterial data of synthesized thioureido derivatives
by: Abdul Kadir, Maisara, et al.
Published: (2019)
by: Abdul Kadir, Maisara, et al.
Published: (2019)
An efficient synthesis of 2,4,7-trisubstituted pyrimido[1,2-a][1,3,5]triazin-6-ones
by: Sachdeva, N., et al.
Published: (2015)
by: Sachdeva, N., et al.
Published: (2015)
Synthesis and Photochemical Properties of Re(I) Tricarbonyl Complexes Bound to Thione and Thiazol-2-ylidene Ligands
by: Stout, Matthew J., et al.
Published: (2020)
by: Stout, Matthew J., et al.
Published: (2020)
Antibacterial and antibiofilm properties of ZnO nanoparticles synthesis using gum arabic as a potential new generation antibacterial agent
by: Norlin, Pauzi, et al.
Published: (2020)
by: Norlin, Pauzi, et al.
Published: (2020)
Molecular docking analysis of Carica papaya Linn constituents as antiviral agent
by: Narayanaswamy, Radhakrishnan, et al.
Published: (2017)
by: Narayanaswamy, Radhakrishnan, et al.
Published: (2017)
Synthesis, spectroscopic studies and antibacterial activity of new lauroyl thiourea amino acid derivatives
by: Abdul Kadir, Maisara, et al.
Published: (2016)
by: Abdul Kadir, Maisara, et al.
Published: (2016)
Synthesis, antiphospholipase A2, antiprotease, antibacterial evaluation and molecular docking analysis of certain novel hydrazones
by: El-Sayed, Nahed Nasser Eid, et al.
Published: (2016)
by: El-Sayed, Nahed Nasser Eid, et al.
Published: (2016)
Self-polymerization of dopamine-coated zinc oxide as a potential antibacterial nanoparticle with molecular docking analysis
by: Albarqouni, Yasin M.Y., et al.
Published: (2025)
by: Albarqouni, Yasin M.Y., et al.
Published: (2025)
Gum arabic as natural stabilizing agent in green synthesis of ZnO nanofluids
for antibacterial application
by: Norlin, Pauzi, et al.
Published: (2019)
by: Norlin, Pauzi, et al.
Published: (2019)
Antibacterial activities of protein extracts from andrographis paniculata, tinospora crispa and centella asiatica
by: Md Zin, Noor Hasniza, et al.
Published: (2016)
by: Md Zin, Noor Hasniza, et al.
Published: (2016)
Antibacterial antivities of protein extracts from Andrographis paniculata, Tinospora crispa and Centella asiatica
by: Md Zin, Noor Hasniza, et al.
Published: (2016)
by: Md Zin, Noor Hasniza, et al.
Published: (2016)
Identifying catalytic residues for peptidases: in silico perspective
by: Muhamad Bunnori, Noraslinda
Published: (2011)
by: Muhamad Bunnori, Noraslinda
Published: (2011)
Identification and characterization of Burkholderia pseudomallei serine and metallopeptidases
by: Muhamad Bunnori, Noraslinda
Published: (2011)
by: Muhamad Bunnori, Noraslinda
Published: (2011)
Potential of Malaysian local honey as an antibacterial agent
by: Ainul Hafiza , A.H., et al.
Published: (2005)
by: Ainul Hafiza , A.H., et al.
Published: (2005)
Synthesis, Characterisation And Molecular Docking Of Quinoxaline-isoxazole Hybrids As Potential Anti-hyperglycemic Agent
by: Phongphane, Lacksany
Published: (2024)
by: Phongphane, Lacksany
Published: (2024)
Molecular docking
by: Abduallah Alsafi, Hassen Mohammed, et al.
Published: (2011)
by: Abduallah Alsafi, Hassen Mohammed, et al.
Published: (2011)
Evaluation of Glass Ionomer Cements
(GICS) properties with coumarin derivatives as
antibacterial agent
by: Mohamad, Dasmawati
Published: (2017)
by: Mohamad, Dasmawati
Published: (2017)
Role of pH on zinc oxide nanoparticles synthesis using gum arabic for sustainable and safe antibacterial agent
by: Norlin, Pauzi, et al.
Published: (2019)
by: Norlin, Pauzi, et al.
Published: (2019)
Potential Of Garcia Mangostana (Mangosteen) Leaves As An Antibacterial Agent
by: Abd Wahab, Mohd Shukor, et al.
Published: (2020)
by: Abd Wahab, Mohd Shukor, et al.
Published: (2020)
Exploit of Malaysian mango kernel extract as antibacterial agent
by: Mirghani, Mohamed Elwathig Saeed, et al.
Published: (2011)
by: Mirghani, Mohamed Elwathig Saeed, et al.
Published: (2011)
Isatin endowed metal chelates as antibacterial and antifungal agents
by: Khalid, Seher, et al.
Published: (2020)
by: Khalid, Seher, et al.
Published: (2020)
Synthesis of ZnO nanoparticles with chitosan as stabilizing agent and their antibacterial properties against Gram-positive and Gram-negative bacteria
by: Nurul Amira, Ahmad Yusof, et al.
Published: (2018)
by: Nurul Amira, Ahmad Yusof, et al.
Published: (2018)
Docking Of Protein With Flavonoids.
by: Ng, Pei Ling, et al.
Published: (2003)
by: Ng, Pei Ling, et al.
Published: (2003)
Crystal structures and docking studies in cathepsin S of bioactive 1,3‐diphenyl‐4‐(trichloro‐λ4‐tellanyl)but‐2‐en‐1‐one derivatives
by: Maganhi, Stella H., et al.
Published: (2021)
by: Maganhi, Stella H., et al.
Published: (2021)
Molecular docking and molecular dynamic simulation of 1,3-Benzoxazine derivatives against penicillin binding protein 2A of methicillin-resistant Staphlyococcus aureus
by: Alharbi, Nourah Jamaan H
Published: (2023)
by: Alharbi, Nourah Jamaan H
Published: (2023)
Synthesis And Characterization Of 1,3-
Disubstituted Benzimidazolium Salts
And Silver(I)-7v-Heterocyclic Carbene
Complexes As Potential Ionic Liquid
Crystals And Antibacterial Agents
by: Yeap, Choon Wan
Published: (2019)
by: Yeap, Choon Wan
Published: (2019)
The potential of sugarcane bagasse as antibacterial agent / Muhammad Syafiq Kamaruzaman
by: Kamaruzaman, Muhammad Syafiq
Published: (2018)
by: Kamaruzaman, Muhammad Syafiq
Published: (2018)
Similar Items
-
Synthesis and molecular docking of 2,4,5-trisubstituted- 1,3-thiazole derivatives as antibacterial agents = Sintesis dan penyatuan molekul terbitan 1,3-tiazol berpenggantian-2,4,5 sebagai agen antibakteria
by: Abdullah Ripain, Iswatun Hasanah, et al.
Published: (2019) -
New 2,4,5-trisubstituted-1,3-thiazole derivatives: synthesis, in vitro antimicrobial activity and in silico study
by: Abdullah Ripain, Iswatun Hasanah, et al.
Published: (2020) -
Design, synthesis and characterization of 2,4-disubstituted-1,3 thiazole amino acid derivatives towards its applications on antimicrobial and antioxidant activities
by: Ngah, Nurziana, et al.
Published: (2018) -
Wound Healing Activity of Pyrazole-thiazole Derivatives of Curcumin Through the Docking, Pharmacokinetics, MD Simulation and MM/GBSA Approaches
by: Forid, Md Shaekh, et al.
Published: (2024) -
Synthesis and molecular docking of carvone derivatives as a potential neuraminidase inhibitors
by: Jusoh, Noorakmar, et al.
Published: (2016)