New quinoxalinone inhibitors targeting secreted phospholipase A2 and alpha-glucosidase

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New quinoxalinone inhibitors targeting secreted phospholipase A2 and alpha-glucosidase

Elevated blood glucose and increased activities of secreted phospholipase A2 (sPLA2) are strongly linked to coronary heart disease. In this report, our goal was to develop small heterocyclic compound that inhibit sPLA2. The title compounds were also tested against α-glucosidase and α-amylase. This a...

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Bibliographic Details
Main Authors:	Alasmary, Fatmah A.S., Alnahdi, Fatima S., Ben Bacha, Abir G., El-Araby, Amr M., Moubayed, Nadine Ms, Alafeefy, Ahmed Mahmoud, El-Araby, Moustafa E.
Format:	Article
Language:	English English
Published:	Informa Healthcare 2017
Subjects:	Q Science (General) QD Chemistry RS Pharmacy and materia medica
Online Access:	http://irep.iium.edu.my/62986/ http://irep.iium.edu.my/62986/2/62986_New%20quinoxalinone%20inhibitors%20targeting%20secreted_scopus.pdf http://irep.iium.edu.my/62986/13/62986_New%20quinoxalinone%20inhibitors.pdf

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