Effect of process variables on the preparation of BSA loaded double-walled poly(lactide-co-glycolide) microspheres

Biodegradable poly(lactide-co-glycolide) (PLGA) microspheres have received much attention over the last twenty-five years for controlled parenteral delivery of therapeutic protein and peptide drugs [1, 2]. In general, for protein drugs delivery, PLGA and PLGA-based single-polymer microspheres system...

Full description

Bibliographic Details
Main Authors: Rahman, Md. Mokhlesur, Ansary, R.H., Mohamed, Farahidah, Kasmuri, Abdul Razak, Md Aris, Mohd Aznan, Katas, H, Awang, M.B.
Format: Proceeding Paper
Language:English
English
Published: 2016
Subjects:
Online Access:http://irep.iium.edu.my/52222/
http://irep.iium.edu.my/52222/2/participation%20Cert.%20scan.jpg
http://irep.iium.edu.my/52222/13/52222.pdf
_version_ 1848784018035703808
author Rahman, Md. Mokhlesur
Ansary, R.H.
Mohamed, Farahidah
Kasmuri, Abdul Razak
Md Aris, Mohd Aznan
Katas, H
Awang, M.B.
author_facet Rahman, Md. Mokhlesur
Ansary, R.H.
Mohamed, Farahidah
Kasmuri, Abdul Razak
Md Aris, Mohd Aznan
Katas, H
Awang, M.B.
author_sort Rahman, Md. Mokhlesur
building IIUM Repository
collection Online Access
description Biodegradable poly(lactide-co-glycolide) (PLGA) microspheres have received much attention over the last twenty-five years for controlled parenteral delivery of therapeutic protein and peptide drugs [1, 2]. In general, for protein drugs delivery, PLGA and PLGA-based single-polymer microspheres system still suffer from two major technical problems associated with their inherent stability problem [3]. Initial burst release followed by very slow and incomplete release is one of the most serious problems in the formulation of PLGA-based protein drugs delivery system. Many strategies have been explored currently to reduce the high initial burst release of protein and peptide drugs from PLGA microspheres [4]. Fabrication of double-walled microspheres in which protein drugs encapsulated in the inner core surrounded by a drug free outer polymer layer offers a promising technique in reducing the high initial burst release. In previous studies, large size double-walled microspheres have been prepared using poly(L-lactic acid) (PLLA) and different co-polymers of PLGA (ester-terminated and carboxyl-terminated) as the core and shell material. Double-walled microspheres consisting PLLA and ester-terminated PLGA as the core or shell material required more time for the complete release of encapsulated drugs due to the slow degrading nature of these polymers.
first_indexed 2025-11-14T16:30:34Z
format Proceeding Paper
id iium-52222
institution International Islamic University Malaysia
institution_category Local University
language English
English
last_indexed 2025-11-14T16:30:34Z
publishDate 2016
recordtype eprints
repository_type Digital Repository
spelling iium-522222022-07-07T07:13:05Z http://irep.iium.edu.my/52222/ Effect of process variables on the preparation of BSA loaded double-walled poly(lactide-co-glycolide) microspheres Rahman, Md. Mokhlesur Ansary, R.H. Mohamed, Farahidah Kasmuri, Abdul Razak Md Aris, Mohd Aznan Katas, H Awang, M.B. QD Chemistry Biodegradable poly(lactide-co-glycolide) (PLGA) microspheres have received much attention over the last twenty-five years for controlled parenteral delivery of therapeutic protein and peptide drugs [1, 2]. In general, for protein drugs delivery, PLGA and PLGA-based single-polymer microspheres system still suffer from two major technical problems associated with their inherent stability problem [3]. Initial burst release followed by very slow and incomplete release is one of the most serious problems in the formulation of PLGA-based protein drugs delivery system. Many strategies have been explored currently to reduce the high initial burst release of protein and peptide drugs from PLGA microspheres [4]. Fabrication of double-walled microspheres in which protein drugs encapsulated in the inner core surrounded by a drug free outer polymer layer offers a promising technique in reducing the high initial burst release. In previous studies, large size double-walled microspheres have been prepared using poly(L-lactic acid) (PLLA) and different co-polymers of PLGA (ester-terminated and carboxyl-terminated) as the core and shell material. Double-walled microspheres consisting PLLA and ester-terminated PLGA as the core or shell material required more time for the complete release of encapsulated drugs due to the slow degrading nature of these polymers. 2016 Proceeding Paper NonPeerReviewed application/pdf en http://irep.iium.edu.my/52222/2/participation%20Cert.%20scan.jpg application/pdf en http://irep.iium.edu.my/52222/13/52222.pdf Rahman, Md. Mokhlesur and Ansary, R.H. and Mohamed, Farahidah and Kasmuri, Abdul Razak and Md Aris, Mohd Aznan and Katas, H and Awang, M.B. (2016) Effect of process variables on the preparation of BSA loaded double-walled poly(lactide-co-glycolide) microspheres. In: International Conference on Industrial Pharmacy (2nd ICIP 2016), 15th-16th Aug. 2016, Kuantan, Pahang. (Unpublished)
spellingShingle QD Chemistry
Rahman, Md. Mokhlesur
Ansary, R.H.
Mohamed, Farahidah
Kasmuri, Abdul Razak
Md Aris, Mohd Aznan
Katas, H
Awang, M.B.
Effect of process variables on the preparation of BSA loaded double-walled poly(lactide-co-glycolide) microspheres
title Effect of process variables on the preparation of BSA loaded double-walled poly(lactide-co-glycolide) microspheres
title_full Effect of process variables on the preparation of BSA loaded double-walled poly(lactide-co-glycolide) microspheres
title_fullStr Effect of process variables on the preparation of BSA loaded double-walled poly(lactide-co-glycolide) microspheres
title_full_unstemmed Effect of process variables on the preparation of BSA loaded double-walled poly(lactide-co-glycolide) microspheres
title_short Effect of process variables on the preparation of BSA loaded double-walled poly(lactide-co-glycolide) microspheres
title_sort effect of process variables on the preparation of bsa loaded double-walled poly(lactide-co-glycolide) microspheres
topic QD Chemistry
url http://irep.iium.edu.my/52222/
http://irep.iium.edu.my/52222/2/participation%20Cert.%20scan.jpg
http://irep.iium.edu.my/52222/13/52222.pdf