Molecular Dynamics Simulation of the Permeation of Lipid- Conjugated Peptides through the Stratum Corneum

This thesis presents a significant advance in selection of drug candidates for transdermal drug delivery. The methodology uses molecular dynamics simulations to understand the translocation of drug candidates across a model of the skin barrier, in atomistic detail. With this, researchers can predict...

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Bibliographic Details
Main Author: Ruiz Perez, Lanie
Format: Thesis
Published: Curtin University 2021
Online Access:http://hdl.handle.net/20.500.11937/87911
Description
Summary:This thesis presents a significant advance in selection of drug candidates for transdermal drug delivery. The methodology uses molecular dynamics simulations to understand the translocation of drug candidates across a model of the skin barrier, in atomistic detail. With this, researchers can predict the translocation rate and efficiently shortlist the drug candidates before conducting costly laboratory-based trials. More importantly, predictions are made with high confidence due to the clarification of the molecular mechanism of translocation.