Design, synthesis, and biological evaluation of novel arylcarboxamide derivatives as anti-tubercular agents
Our group has previously reported several indolecarboxamides exhibiting potent antitubercular activity. Herein, we rationally designed several arylcarboxamides based on our previously reported homology model and the recently published crystal structure of the mycobacterial membrane protein large 3 (...
| Main Authors: | Alsayed, Shahinda SR, Lun, Shichun, Luna, Giuseppe, Beh, Chau Chun, Payne, Alan D, Foster, Neil R, Bishai, William R, Gunosewoyo, Hendra |
|---|---|
| Format: | Journal Article |
| Published: |
RSC
2020
|
| Online Access: | http://purl.org/au-research/grants/arc/DE160100482 http://hdl.handle.net/20.500.11937/78250 |
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