A one-pot, three-component aminotriazine annulation onto 5-aminopyrazole-4-carbonitriles under microwave irradiation

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A one-pot, three-component aminotriazine annulation onto 5-aminopyrazole-4-carbonitriles under microwave irradiation

A one-pot, three-component, microwave-assisted reaction of 5-aminopyrazole-4-carbonitriles, triethyl orthoformate and cyanamide afforded novel 7-arylamino-substituted 4-aminopyrazolo[1,5-a][1,3,5]triazine-8-carbonitriles. The reaction proceeded in a chemo- and regioselective manner resulting in the...

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Bibliographic Details
Main Authors:	Lim, Felicia Phei Lin, Luna, Giuseppe, Dolzhenko, Anton
Format:	Journal Article
Published:	Pergamon 2015
Subjects:	Purine isostere Multicomponent reaction Microwave-assisted synthesis Triazine Pyrazole
Online Access:	http://hdl.handle.net/20.500.11937/5411

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