Role of NF-κB in tumorigenesis

Persistent activation of the pro-inflammatory transcription factor nuclear factor-κB (NF-κB) is frequently observed in several human malignancies and can drive the processes of tumor initiation, oncogenic transformation, and malignant progression. Once activated, this master transcription factor reg...

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Main Authors: Shanmugam, M., Kumar, Alan Prem, Tan, B., Sethi, G.
Format: Journal Article
Published: 2013
Online Access:http://hdl.handle.net/20.500.11937/53174
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author Shanmugam, M.
Kumar, Alan Prem
Tan, B.
Sethi, G.
author_facet Shanmugam, M.
Kumar, Alan Prem
Tan, B.
Sethi, G.
author_sort Shanmugam, M.
building Curtin Institutional Repository
collection Online Access
description Persistent activation of the pro-inflammatory transcription factor nuclear factor-κB (NF-κB) is frequently observed in several human malignancies and can drive the processes of tumor initiation, oncogenic transformation, and malignant progression. Once activated, this master transcription factor regulates the expression of numerous genes involved in proliferation, survival, metastasis, angiogenesis, chemoresistance, and radioresistance. Thus, novel pharmacological agents that can suppress constitutive and/or inducible NF-κB activation have the potential for cancer therapy. In this review, we describe in detail the pleiotropic molecular mechanisms of aberrant NF-κB activation and also discuss various therapeutic strategies employed to suppress deregulated activation of this important oncogenic transcription factor in cancer.
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spelling curtin-20.500.11937-531742017-10-12T06:06:19Z Role of NF-κB in tumorigenesis Shanmugam, M. Kumar, Alan Prem Tan, B. Sethi, G. Persistent activation of the pro-inflammatory transcription factor nuclear factor-κB (NF-κB) is frequently observed in several human malignancies and can drive the processes of tumor initiation, oncogenic transformation, and malignant progression. Once activated, this master transcription factor regulates the expression of numerous genes involved in proliferation, survival, metastasis, angiogenesis, chemoresistance, and radioresistance. Thus, novel pharmacological agents that can suppress constitutive and/or inducible NF-κB activation have the potential for cancer therapy. In this review, we describe in detail the pleiotropic molecular mechanisms of aberrant NF-κB activation and also discuss various therapeutic strategies employed to suppress deregulated activation of this important oncogenic transcription factor in cancer. 2013 Journal Article http://hdl.handle.net/20.500.11937/53174 10.1615/ForumImmunDisTher.2013008382 restricted
spellingShingle Shanmugam, M.
Kumar, Alan Prem
Tan, B.
Sethi, G.
Role of NF-κB in tumorigenesis
title Role of NF-κB in tumorigenesis
title_full Role of NF-κB in tumorigenesis
title_fullStr Role of NF-κB in tumorigenesis
title_full_unstemmed Role of NF-κB in tumorigenesis
title_short Role of NF-κB in tumorigenesis
title_sort role of nf-κb in tumorigenesis
url http://hdl.handle.net/20.500.11937/53174