A new, one-pot, multicomponent synthesis of 5-aza-9-deaza-adenines under microwave irradiation

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A new, one-pot, multicomponent synthesis of 5-aza-9-deaza-adenines under microwave irradiation

A new, practical, three-component method for the synthesis of 5-aza-9-deaza-adenines is developed. Aminopyrazoles react in a one-pot fashion with triethyl orthoformate and cyanamide under microwave irradiation affording 5-aza-9-deaza-adenines in good yields and high purity. The main advantages of th...

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Bibliographic Details
Main Authors:	Lim, Felicia Phei Lin, Luna, Giuseppe, Dolzhenko, Anton
Format:	Journal Article
Published:	Pergamon 2014
Subjects:	Cyanamide Multicomponent reaction Triazine Pyrazole Purine analogue
Online Access:	http://hdl.handle.net/20.500.11937/44673

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