Acyl lipidation of a peptide: effects on activity and epidermal permeability in vitro

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Acyl lipidation of a peptide: effects on activity and epidermal permeability in vitro

Short-chain lipid conjugates can increase permeability of a small peptide across human epidermis; however, the emerging lipoaminoacid (LAA) conjugation technique is costly and can deliver mixed synthetic products of varied biological potential. LAA conjugation using a racemic mixture produces a mixt...

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Bibliographic Details
Main Authors:	Rocco, D., Ross, J., Murray, P., Caccetta, Rima
Format:	Journal Article
Published:	Dove Medical Press Ltd. 2016
Online Access:	http://hdl.handle.net/20.500.11937/40778

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