A novel folic acid-conjugated TiO2–SiO2 photosensitizer for cancer targeting in photodynamic therapy

In this paper, a novel folic acid-conjugated silica-coated titanium dioxide (TiO2–SiO2) photosensitizer was synthesized and characterized using various analytical instruments. The photosensitizer was further assessed with regards to its photoreactivity, cellular and hemocompatibility, cell internali...

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Main Authors: Feng, Xiaohui, Zhang, S., Wu, H., Lou, Xia
Format: Journal Article
Published: Elsevier BV 2015
Subjects:
Online Access:http://hdl.handle.net/20.500.11937/37859
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author Feng, Xiaohui
Zhang, S.
Wu, H.
Lou, Xia
author_facet Feng, Xiaohui
Zhang, S.
Wu, H.
Lou, Xia
author_sort Feng, Xiaohui
building Curtin Institutional Repository
collection Online Access
description In this paper, a novel folic acid-conjugated silica-coated titanium dioxide (TiO2–SiO2) photosensitizer was synthesized and characterized using various analytical instruments. The photosensitizer was further assessed with regards to its photoreactivity, cellular and hemocompatibility, cell internalization, and phototoxicity. Conjugating folic acid with TiO2–SiO2 has shown a significantly improved compatibility of the nanoparticles with the mouse fibroblast cells (L929) at 24 h. An improved compatibility with the human nasopharyngeal epidermoid cancer (KB) cells was also demonstrated, but to a slightly reduced degree. Enhanced cell internalization was well demonstrated in the TiO2–SiO2 folate nanoparticles. Upon exposure to UV light, TiO2–SiO2 folate nanoparticles maintained a high level photodynamic reactivity and yielded a 38–43% photo-killing of KB cells. The photo-killing effect increased with increasing dosage in the investigated concentration range of 50–100 μg ml−1.
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publishDate 2015
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spelling curtin-20.500.11937-378592017-09-13T15:58:42Z A novel folic acid-conjugated TiO2–SiO2 photosensitizer for cancer targeting in photodynamic therapy Feng, Xiaohui Zhang, S. Wu, H. Lou, Xia Photodynamic therapy Photo-killing Titanium dioxide nanoparticles Photosensitizer Folic acid Targeting In this paper, a novel folic acid-conjugated silica-coated titanium dioxide (TiO2–SiO2) photosensitizer was synthesized and characterized using various analytical instruments. The photosensitizer was further assessed with regards to its photoreactivity, cellular and hemocompatibility, cell internalization, and phototoxicity. Conjugating folic acid with TiO2–SiO2 has shown a significantly improved compatibility of the nanoparticles with the mouse fibroblast cells (L929) at 24 h. An improved compatibility with the human nasopharyngeal epidermoid cancer (KB) cells was also demonstrated, but to a slightly reduced degree. Enhanced cell internalization was well demonstrated in the TiO2–SiO2 folate nanoparticles. Upon exposure to UV light, TiO2–SiO2 folate nanoparticles maintained a high level photodynamic reactivity and yielded a 38–43% photo-killing of KB cells. The photo-killing effect increased with increasing dosage in the investigated concentration range of 50–100 μg ml−1. 2015 Journal Article http://hdl.handle.net/20.500.11937/37859 10.1016/j.colsurfb.2014.11.035 Elsevier BV fulltext
spellingShingle Photodynamic therapy
Photo-killing
Titanium dioxide nanoparticles
Photosensitizer
Folic acid
Targeting
Feng, Xiaohui
Zhang, S.
Wu, H.
Lou, Xia
A novel folic acid-conjugated TiO2–SiO2 photosensitizer for cancer targeting in photodynamic therapy
title A novel folic acid-conjugated TiO2–SiO2 photosensitizer for cancer targeting in photodynamic therapy
title_full A novel folic acid-conjugated TiO2–SiO2 photosensitizer for cancer targeting in photodynamic therapy
title_fullStr A novel folic acid-conjugated TiO2–SiO2 photosensitizer for cancer targeting in photodynamic therapy
title_full_unstemmed A novel folic acid-conjugated TiO2–SiO2 photosensitizer for cancer targeting in photodynamic therapy
title_short A novel folic acid-conjugated TiO2–SiO2 photosensitizer for cancer targeting in photodynamic therapy
title_sort novel folic acid-conjugated tio2–sio2 photosensitizer for cancer targeting in photodynamic therapy
topic Photodynamic therapy
Photo-killing
Titanium dioxide nanoparticles
Photosensitizer
Folic acid
Targeting
url http://hdl.handle.net/20.500.11937/37859