Viability and topographical analysis of microencapsulated ß-cells exposed to a biotransformed tertiary bile acid: An ex vivo study

Microencapsulated pancreatic ß-cells have been studied as an ideal system for delivering insulin. However, the clinical applications have not been achieved. We tried multiple excipients/ratios and various methods for producing suitable microcapsules, but success remains limited. A recent study used...

Full description

Bibliographic Details
Main Authors: Mooranian, Armin, Negrulj, Rebecca, Al-Salami, Hani
Format: Journal Article
Published: 2016
Online Access:http://hdl.handle.net/20.500.11937/32621
_version_ 1848753713519263744
author Mooranian, Armin
Negrulj, Rebecca
Al-Salami, Hani
author_facet Mooranian, Armin
Negrulj, Rebecca
Al-Salami, Hani
author_sort Mooranian, Armin
building Curtin Institutional Repository
collection Online Access
description Microencapsulated pancreatic ß-cells have been studied as an ideal system for delivering insulin. However, the clinical applications have not been achieved. We tried multiple excipients/ratios and various methods for producing suitable microcapsules, but success remains limited. A recent study used the tertiary bile acid, taurocholic acid (TCA), to improve the rectal delivery of insulin while another study used TCA to improve the oral delivery of heparin. Thus, in this study, we used TCA in different formulations, using a new microencapsulating method, to study its suitability for ß-cell microencapsulation. Using a methodology at set temperature of 37°C, amplitude of 1.5 and a total gelation time of 21 minutes, ten different formulations were examined (with or without TCA) and all formulations showed similar cell viability, which was enhanced by TCA addition. This suggests potential benefits of our microencapsulating parameters and TCA in ß-cells microencapsulation.
first_indexed 2025-11-14T08:28:53Z
format Journal Article
id curtin-20.500.11937-32621
institution Curtin University Malaysia
institution_category Local University
last_indexed 2025-11-14T08:28:53Z
publishDate 2016
recordtype eprints
repository_type Digital Repository
spelling curtin-20.500.11937-326212017-09-13T15:25:11Z Viability and topographical analysis of microencapsulated ß-cells exposed to a biotransformed tertiary bile acid: An ex vivo study Mooranian, Armin Negrulj, Rebecca Al-Salami, Hani Microencapsulated pancreatic ß-cells have been studied as an ideal system for delivering insulin. However, the clinical applications have not been achieved. We tried multiple excipients/ratios and various methods for producing suitable microcapsules, but success remains limited. A recent study used the tertiary bile acid, taurocholic acid (TCA), to improve the rectal delivery of insulin while another study used TCA to improve the oral delivery of heparin. Thus, in this study, we used TCA in different formulations, using a new microencapsulating method, to study its suitability for ß-cell microencapsulation. Using a methodology at set temperature of 37°C, amplitude of 1.5 and a total gelation time of 21 minutes, ten different formulations were examined (with or without TCA) and all formulations showed similar cell viability, which was enhanced by TCA addition. This suggests potential benefits of our microencapsulating parameters and TCA in ß-cells microencapsulation. 2016 Journal Article http://hdl.handle.net/20.500.11937/32621 10.1504/IJNBM.2016.079684 restricted
spellingShingle Mooranian, Armin
Negrulj, Rebecca
Al-Salami, Hani
Viability and topographical analysis of microencapsulated ß-cells exposed to a biotransformed tertiary bile acid: An ex vivo study
title Viability and topographical analysis of microencapsulated ß-cells exposed to a biotransformed tertiary bile acid: An ex vivo study
title_full Viability and topographical analysis of microencapsulated ß-cells exposed to a biotransformed tertiary bile acid: An ex vivo study
title_fullStr Viability and topographical analysis of microencapsulated ß-cells exposed to a biotransformed tertiary bile acid: An ex vivo study
title_full_unstemmed Viability and topographical analysis of microencapsulated ß-cells exposed to a biotransformed tertiary bile acid: An ex vivo study
title_short Viability and topographical analysis of microencapsulated ß-cells exposed to a biotransformed tertiary bile acid: An ex vivo study
title_sort viability and topographical analysis of microencapsulated ß-cells exposed to a biotransformed tertiary bile acid: an ex vivo study
url http://hdl.handle.net/20.500.11937/32621