Amino acid bioconjugation via iClick reaction of an oxanorbornadiene-masked alkyne with a MnI(bpy)(CO)3-coordinated azide

The catalyst-free room temperature iClick reaction of an unsymmetrically 2,3-disubstituted oxanorbornadiene (OND) as a “masked” alkyne equivalent with [Mn(N3)(bpyCH3,CH3)(CO)3] leads to isolation of a phenylalanine ester bioconjugate, in which the model amino acid is linked to the metal moiety via a...

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Main Authors: Henry, L., Schneider, C., Mützel, B., Simpson, Peter, Nagel, C., Fucke, K., Schatzschneider, U.
Format: Journal Article
Published: 2014
Online Access:http://hdl.handle.net/20.500.11937/21454
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author Henry, L.
Schneider, C.
Mützel, B.
Simpson, Peter
Nagel, C.
Fucke, K.
Schatzschneider, U.
author_facet Henry, L.
Schneider, C.
Mützel, B.
Simpson, Peter
Nagel, C.
Fucke, K.
Schatzschneider, U.
author_sort Henry, L.
building Curtin Institutional Repository
collection Online Access
description The catalyst-free room temperature iClick reaction of an unsymmetrically 2,3-disubstituted oxanorbornadiene (OND) as a “masked” alkyne equivalent with [Mn(N3)(bpyCH3,CH3)(CO)3] leads to isolation of a phenylalanine ester bioconjugate, in which the model amino acid is linked to the metal moiety via a N-2-coordinated triazolate formed in a cycloaddition-retro-Diels–Alder (crDA) reaction sequence, in a novel approach to bioorthogonal coupling reactions based on metal-centered reactivity.
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institution Curtin University Malaysia
institution_category Local University
last_indexed 2025-11-14T07:39:19Z
publishDate 2014
recordtype eprints
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spelling curtin-20.500.11937-214542018-03-29T09:06:35Z Amino acid bioconjugation via iClick reaction of an oxanorbornadiene-masked alkyne with a MnI(bpy)(CO)3-coordinated azide Henry, L. Schneider, C. Mützel, B. Simpson, Peter Nagel, C. Fucke, K. Schatzschneider, U. The catalyst-free room temperature iClick reaction of an unsymmetrically 2,3-disubstituted oxanorbornadiene (OND) as a “masked” alkyne equivalent with [Mn(N3)(bpyCH3,CH3)(CO)3] leads to isolation of a phenylalanine ester bioconjugate, in which the model amino acid is linked to the metal moiety via a N-2-coordinated triazolate formed in a cycloaddition-retro-Diels–Alder (crDA) reaction sequence, in a novel approach to bioorthogonal coupling reactions based on metal-centered reactivity. 2014 Journal Article http://hdl.handle.net/20.500.11937/21454 10.1039/c4cc07892f restricted
spellingShingle Henry, L.
Schneider, C.
Mützel, B.
Simpson, Peter
Nagel, C.
Fucke, K.
Schatzschneider, U.
Amino acid bioconjugation via iClick reaction of an oxanorbornadiene-masked alkyne with a MnI(bpy)(CO)3-coordinated azide
title Amino acid bioconjugation via iClick reaction of an oxanorbornadiene-masked alkyne with a MnI(bpy)(CO)3-coordinated azide
title_full Amino acid bioconjugation via iClick reaction of an oxanorbornadiene-masked alkyne with a MnI(bpy)(CO)3-coordinated azide
title_fullStr Amino acid bioconjugation via iClick reaction of an oxanorbornadiene-masked alkyne with a MnI(bpy)(CO)3-coordinated azide
title_full_unstemmed Amino acid bioconjugation via iClick reaction of an oxanorbornadiene-masked alkyne with a MnI(bpy)(CO)3-coordinated azide
title_short Amino acid bioconjugation via iClick reaction of an oxanorbornadiene-masked alkyne with a MnI(bpy)(CO)3-coordinated azide
title_sort amino acid bioconjugation via iclick reaction of an oxanorbornadiene-masked alkyne with a mni(bpy)(co)3-coordinated azide
url http://hdl.handle.net/20.500.11937/21454