Search Results - Stocks, Michael

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  1. 1
    Ipratropium is ‘luminally recycled’ by an inter-play between apical uptake and efflux transporters in Calu-3 bronchial epithelial cell layers

    Ipratropium is ‘luminally recycled’ by an inter-play between apical uptake and efflux transporters in Calu-3 bronchial epithelial cell layers by Panduga, Vijender, Stocks, Michael J., Bosquillon, Cynthia

    Published 2017
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  2. 2
    Drug-like antagonists of P2Y receptors — from lead identification to drug development

    Drug-like antagonists of P2Y receptors — from lead identification to drug development by Conroy, Sean, Kindon, Nicholas, Kellam, Barrie, Stocks, Michael

    Published 2016
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  3. 3
    Pseudomonas aeruginosa quorum sensing systems as drug discovery targets: current position and future perspectives

    Pseudomonas aeruginosa quorum sensing systems as drug discovery targets: current position and future perspectives by Soukarieh, Fadi, Williams, Paul, Stocks, Michael John, Camara, Miguel

    Published 2018
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  4. 4
    Synthesis of new DPP-4 inhibitors based on a novel tricyclic scaffold

    Synthesis of new DPP-4 inhibitors based on a novel tricyclic scaffold by Schwehm, Carolin, Li, Jin, Song, Hongmei, Hu, Xiao, Kellam, Barrie, Stocks, Michael

    Published 2015
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  5. 5
    Preparation and structural analysis of (±)-cis-ethyl 2-sulfanylidenedecahydro-1,6-naphthyridine-6-carboxylate and (±)-trans-ethyl 2-oxooctahydro-1H-pyrrolo[3,2-c]pyridine-5-carboxylate

    Preparation and structural analysis of (±)-cis-ethyl 2-sulfanylidenedecahydro-1,6-naphthyridine-6-carboxylate and (±)-trans-ethyl 2-oxooctahydro-1H-pyrrolo[3,2-c]pyridine-5-carboxy... by Schwehm, Carolin, Lewis, William, Blake, Alexander J., Kellam, Barrie, Stocks, Michael J.

    Published 2014
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  6. 6
    Linifanib – a multi-targeted receptor tyrosine kinase inhibitor and a low molecular weight gelator

    Linifanib – a multi-targeted receptor tyrosine kinase inhibitor and a low molecular weight gelator by Marlow, Maria, Al-Ameedee, Mohammed, Smith, Thomas, Wheeler, Simon, Stocks, Michael J.

    Published 2015
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  7. 7
    Nucleoside based self-assembling drugs for localized drug delivery

    Nucleoside based self-assembling drugs for localized drug delivery by Skilling, Kathryn J., Stocks, Michael J., Kellam, Barrie, Ashford, Marianne, Bradshaw, Tracey, Burroughs, Laurence, Marlow, Maria

    Published 2018
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  8. 8
    Synthesis and evaluation of the first fluorescent antagonists of the human P2Y2 receptor based on AR-C118925

    Synthesis and evaluation of the first fluorescent antagonists of the human P2Y2 receptor based on AR-C118925 by Conroy, Sean, Kindon, Nicholas, Glenn, Jacqueline, Stoddart, Leigh A., Lewis, Richard James, Hill, Stephen J., Kellam, Barrie, Stocks, Michael J.

    Published 2018
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  9. 9
    From UTP to AR-C118925, the discovery of a potent non nucleotide antagonist of the P2Y2 receptor

    From UTP to AR-C118925, the discovery of a potent non nucleotide antagonist of the P2Y2 receptor by Kindon, Nicholas, Davis, Andrew, Dougall, Iain, Dixon, John, Johnson, Timothy, Walters, Iain, Thom, Steve, McKechnie, Kenneth, Meghani, Premji, Stocks, Michael

    Published 2017
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  10. 10
    Self-assembling benzothiazole-based gelators: a mechanistic understanding of in vitro bioactivation and gelation

    Self-assembling benzothiazole-based gelators: a mechanistic understanding of in vitro bioactivation and gelation by Citossi, Francesca, Smith, Thomas, Lee, Jong Bong, Segal, Joel, Gershkovich, Pavel, Stocks, Michael John, Bradshaw, Tracey D., Kellam, Barrie, Marlow, Maria

    Published 2018
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  11. 11
    Design and elaboration of a tractable tricyclic scaffold to synthesize druglike inhibitors of dipeptidyl peptidase-4 (DPP-4), antagonists of the C–C Chemokine Receptor Type 5 (CCR5), and highly potent and selective phosphoinositol-3 Kinase δ (PI3Kδ) inhibitors

    Design and elaboration of a tractable tricyclic scaffold to synthesize druglike inhibitors of dipeptidyl peptidase-4 (DPP-4), antagonists of the C–C Chemokine Receptor Type 5 (CCR5... by Schwehm, Carolin, Kellam, Barrie, Garces, Aimie, Hill, Stephen J., Kindon, Nicholas, Bradshaw, Tracey D., Li, Jin, Macdonald, Simon J.F., Rowedder, James E., Stoddart, Leigh A., Stocks, Michael

    Published 2017
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  12. 12
    In silico and in vitro-guided identification of inhibitors of alkylquinolone-dependent quorum sensing in Pseudomonas aeruginosa

    In silico and in vitro-guided identification of inhibitors of alkylquinolone-dependent quorum sensing in Pseudomonas aeruginosa by Soukarieh, Fadi, Oton, Eduard Vico, Dubern, Jean-Frédéric, Gomes, Janice, Halliday, Nigel, de Pilar Crespo, Maria, Ramírez-Prada, Jonathan, Insuasty, Braulio, Abonia, Rodrigo, Quiroga, Jairo, Heeb, Stephan, Williams, Paul, Stocks, Michael J., Cámara, Miguel

    Published 2018
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  13. 13
    Discovery of AZD3199, an inhaled ultralong acting β2 receptor agonist with rapid onset of action

    Discovery of AZD3199, an inhaled ultralong acting β2 receptor agonist with rapid onset of action by Stocks, Michael, Alcaraz, Lilian, Bailey, Andrew, Bonnert, Roger, Cadogan, Elaine, Christie, Jadeen, Dixon, John, Connolly, Stephen, Cook, Anthony, Fisher, Adrian, Flaherty, Alice, Humphries, Alexander, Ingall, Anthony, Jordan, Stephen, Lawson, Mandy, Mullen, Alex, Nicholls, David, Paine, Stuart, Pairaudeau, Garry, Young, Alan

    Published 2014
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  14. 14
    Discovery of AZD-2098 and AZD-1678, two potent and bioavailable CCR4 receptor antagonists

    Discovery of AZD-2098 and AZD-1678, two potent and bioavailable CCR4 receptor antagonists by Kindon, Nicholas, Andrews, Glen, Baxter, Andrew, Cheshire, David, Hemsley, Paul, Johnson, Timothy, Liu, Yu-Zhen, McGinnity, Dermot, McHale, Mark, Mete, Antonio, Reuberson, James, Roberts, Bryan, Steele, John, Teobald, Barry, Unitt, John, Vaughan, Deborah, Walters, Iain, Stocks, Michael J.

    Published 2017
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  15. 15
    Lipophilic activated ester prodrug approach for drug delivery to the intestinal lymphatic system

    Lipophilic activated ester prodrug approach for drug delivery to the intestinal lymphatic system by Lee, Jong Bong, Zgair, Atheer, Malec, Jed, Kim, Tae Hwan, Kim, Min Gi, Ali, Joseph, Qin, Chaolong, Feng, Wanshan, Chiang, Manting, Gao, Xizhe, Voronin, Gregory, Garces, Aimie, Lau, Chun Long, Chan, Ting-Hoi, Hume, Amy, McIntosh, Tecashanell M., Soukarieh, Fadi, Al-Hayali, Mohammed, Cipolla, Elena, Collins, Hilary M., Heery, David M., Shin, Beom Soo, Yoo, Sun Dong, Kagan, Leonid, Stocks, Michael J., Bradshaw, Tracey D., Fischer, Peter M., Gershkovich, Pavel

    Published 2018
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