Search Results - Fischer, Peter M.

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  1. 1
    Approved and experimental small-molecule oncology kinase inhibitor drugs: a mid-2016 overview

    Approved and experimental small-molecule oncology kinase inhibitor drugs: a mid-2016 overview by Fischer, Peter M.

    Published 2017
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  2. 2
    Design of small-molecule active-site inhibitors of the S1A family proteases as procoagulant and anticoagulant drugs

    Design of small-molecule active-site inhibitors of the S1A family proteases as procoagulant and anticoagulant drugs by Fischer, Peter M.

    Published 2017
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  3. 3
    A facile approach to tryptophan derivatives for the total synthesis of argyrin analogues

    A facile approach to tryptophan derivatives for the total synthesis of argyrin analogues by Chen, Chou-Hsiung, Genapathy, Sivaneswary, Fischer, Peter M., Chan, Weng C.

    Published 2014
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  4. 4
    Three-dimensional pharmacophore design and biochemical screening identifies substituted 1,2,4-triazoles as inhibitors of the annexin A2-S100A10 protein interaction

    Three-dimensional pharmacophore design and biochemical screening identifies substituted 1,2,4-triazoles as inhibitors of the annexin A2-S100A10 protein interaction by Reddy, Tummala R.K., Li, Chan, Fischer, Peter M., Dekker, Lodewijk V.

    Published 2012
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  5. 5
    Multiple linear regression modelling to predict the stability of polymer-drug solid dispersions: comparison of the effects of polymers and manufacturing methods on solid dispersion stability

    Multiple linear regression modelling to predict the stability of polymer-drug solid dispersions: comparison of the effects of polymers and manufacturing methods on solid dispersion... by Fridgeirsdottir, Gudrun, Harris, Robert, Dryden, Ian L., Fischer, Peter M., Roberts, Clive J.

    Published 2018
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  6. 6
    Design, synthesis and SAR exploration of tri-substituted 1,2,4-triazoles as inhibitors of the annexin A2–S100A10 protein interaction

    Design, synthesis and SAR exploration of tri-substituted 1,2,4-triazoles as inhibitors of the annexin A2–S100A10 protein interaction by Reddy, Tummala R.K., Li, Chan, Guo, Xiaoxia, Fischer, Peter M., Dekker, Lodewijk V.

    Published 2014
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  7. 7
    GPCRs through the keyhole: the role of protein flexibility in ligand binding to β-adrenoceptors

    GPCRs through the keyhole: the role of protein flexibility in ligand binding to β-adrenoceptors by Emtage, Abigail L., Mistry, Shailesh N., Fischer, Peter M., Kellam, Barrie, Laughton, Charles A.

    Published 2016
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  8. 8
    PPP1R15A-mediated dephosphorylation of eIF2α is unaffected by Sephin1 or Guanabenz

    PPP1R15A-mediated dephosphorylation of eIF2α is unaffected by Sephin1 or Guanabenz by Crespillo-Casado, Ana, Chambers, Joseph E., Fischer, Peter M., Marciniak, Stefan J., Ron, David

    Published 2017
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  9. 9
    Assessment of the protein interaction between coagulation factor XII and corn trypsin inhibitor by molecular docking and biochemical validation

    Assessment of the protein interaction between coagulation factor XII and corn trypsin inhibitor by molecular docking and biochemical validation by Hamad, Badraldin K., Pathak, Monika, Manna, Rosa, Fischer, Peter M., Emsley, Jonas, Dekker, Lodewijk V.

    Published 2017
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  10. 10
    Development of cordycepin formulations for preclinical and clinical studies

    Development of cordycepin formulations for preclinical and clinical studies by Lee, Jong Bong, Adrower, Cecilia, Qin, Chaolong, Fischer, Peter M., Moor, Cornelia H. de, Gershkovich, Pavel

    Published 2017
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  11. 11
    Synthesis and in vitro and in vivo characterization of highly β1-Selective β-Adrenoceptor partial agonists

    Synthesis and in vitro and in vivo characterization of highly β1-Selective β-Adrenoceptor partial agonists by Mistry, Shailesh N., Baker, Jillian G., Fischer, Peter M., Hill, Stephen J., Gardiner, Sheila M., Kellam, Barrie

    Published 2013
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  12. 12
    In vitro and in vivo analysis of a novel highly selective β1-adrenoceptor partial agonist.

    In vitro and in vivo analysis of a novel highly selective β1-adrenoceptor partial agonist. by Baker, Jillian G., Mistry, Shailesh N., Fischer, Peter M., Hill, Stephen J., Gardiner, Sheila M., Kellam, Barrie

    Published 2012
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  13. 13
    The Meisenheimer complex as a paradigm in drug discovery: reversible covalent inhibition through C67 of the ATP binding site of PLK1

    The Meisenheimer complex as a paradigm in drug discovery: reversible covalent inhibition through C67 of the ATP binding site of PLK1 by Pearson, Russell J., Blake, David G., Mezna, Mokdad, Fischer, Peter M., Westwood, Nicholas J., McInnes, Campbell

    Published 2018
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  14. 14
    Simple and sensitive HPLC-UV method for determination of bexarotene in rat plasma

    Simple and sensitive HPLC-UV method for determination of bexarotene in rat plasma by Lee, Jong Bong, Zgair, Atheer, Kim, Tae Hwan, Kim, Min Gi, Yoo, Sun Dong, Fischer, Peter M., Gershkovich, Pavel

    Published 2017
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  15. 15
    A fluorescence-based assay suitable for quantitative analysis of deadenylase enzyme activity

    A fluorescence-based assay suitable for quantitative analysis of deadenylase enzyme activity by Maryati, Marayti, Kaur, Ishwinder, Jadhav, Gopal P., Olotu-Umoren, Loyin, Oveh, Blessing, Hashmi, Lubna, Fischer, Peter M., Winkler, G. Sebastiaan

    Published 2013
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  16. 16
    Quantitative analysis of lab-to-lab variability in Caco-2 permeability assays

    Quantitative analysis of lab-to-lab variability in Caco-2 permeability assays by Lee, Jong Bong, Zgair, Atheer, Taha, Dhiaa A., Zang, Xiaowei, Kagan, Leonid, Kim, Tae Hwan, Kim, Min Gi, Yun, Hwi-yeol, Fischer, Peter M., Gershkovich, Pavel

    Published 2017
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  17. 17
    Novel selective β1-adrenoceptor antagonists for concomitant cardiovascular and respiratory disease

    Novel selective β1-adrenoceptor antagonists for concomitant cardiovascular and respiratory disease by Baker, Jillian G., Gardiner, Sheila M., Woolard, Jeanette, Fromont, Christophe, Jadhav, Gopal P., Mistry, Shailesh N., Thompson, Kevin S.J., Kellam, Barrie, Hill, Stephen J., Fischer, Peter M.

    Published 2017
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  18. 18
    Dietary fats and pharmaceutical lipid excipients increase systemic exposure to orally administered cannabis and cannabis-based medicines

    Dietary fats and pharmaceutical lipid excipients increase systemic exposure to orally administered cannabis and cannabis-based medicines by Zgair, Atheer, Wong, Jonathan C.M., Lee, Jong Bong, Mistry, Jatin, Sivak, Olena, Wasan, Kishor M., Hennig, Ivo M., Barrett, David A., Constantinescu, Cris S., Fischer, Peter M., Gershkovich, Pavel

    Published 2016
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  19. 19
    Design of nucleotide-mimetic and non-nucleotide inhibitors of the translation initiation factor eIF4E: synthesis, structural and functional characterisation

    Design of nucleotide-mimetic and non-nucleotide inhibitors of the translation initiation factor eIF4E: synthesis, structural and functional characterisation by Soukarieh, Fadi, Nowicki, Matthew W., Bastide, Amandine, Poyry, Tuija, Jones, Carolyn, Dudek, Kate, Patwardhan, Geetanjali, Meullenet, François, Oldham, Neil J., Walkinshaw, Malcolm D., Willis, Anne E., Fischer, Peter M.

    Published 2016
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  20. 20
    Binding of ISRIB reveals a regulatory site in the nucleotide exchange factor eIF2B

    Binding of ISRIB reveals a regulatory site in the nucleotide exchange factor eIF2B by Zyryanova, Alisa F., Weis, Félix, Faille, Alexandre, Abo Alard, Akeel, Crespillo-Casado, Ana, Sekine, Yusuke, Harding, Heather P., Allen, Felicity, Parts, Leopold, Fromont, Christoph, Fischer, Peter M., Warren, Alan J., Ron, David

    Published 2018
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